Target Details
UniProt ACP31644
Gene SymbolGABRA5
Protein NameGamma-aminobutyric acid receptor subunit alpha-5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,276
  • Clinical molecules 0
  • Avg pChEMBL 7.87
Top Co-occurrence Targets
Active Molecules (1,276)
InChIKey pChEMBL Type Targets Clinical
AWOOMIRCBITDFK 10.0 Ki 6
FNCCIRFBYGUBRQ 10.0 Ki 5
HLKYSQGBIIIQJN 9.9 Ki 5
PEBWTLIJBCZFOA 9.9 Ki 6
IQKMZIHHJYCEKH 9.8 Ki 5
XJRDHPKTMGWJGN 9.8 Ki 6
RUOVJURXWIHZPL 9.8 Ki 5
RYKBQSSZEXHGJL 9.8 Ki 5
MZFKWSFOAVBLQM 9.8 IC50 16
UWXAQZGCSSYTJL 9.8 Ki 6
WDBBCFFNOHDOBT 9.7 Ki 5
ZQLPLWRQUVVKJZ 9.7 Ki 6
GFTZCCLPKHGIAB 9.7 Ki 3
GMFQPQQGURBQLQ 9.7 Ki 3
NVETZYIXXYETLA 9.7 Ki 6
PCLDOYFAYOCLQE 9.7 Ki 3
PPAPIXRCRCPGPU 9.7 Ki 3
QKIWQBLNTSQOLY 9.7 Ki 6
RCZMTZGAJGJJDL 9.7 Ki 3
WFPXOWCKXUEKCA 9.7 IC50 16
WSSWOLULTYVMTE 9.7 Ki 3
YWVNAIWRDXBOOS 9.7 Ki 6
FTBGMXWQYKNAKT 9.7 Ki 6
VYBPWFTWAKMZPZ 9.7 Ki 5
GOIFCXRIFSYPFG 9.6 Ki 5
KVKWRJDNIJTMGN 9.6 IC50 16
JOHKRJNYKDHTID 9.6 Ki 6
MTOXGGJOEHOEJT 9.6 Ki 5
ZRKDDZBVSZLOFS 9.6 Ki 6
QNLKJSGZMGMFBW 9.5 Ki 6
RZOFEWOHNOOHND 9.5 Ki 6
BFKIZTLCAFUHPD 9.5 Ki 2
LCDOZBPYZHDFGO 9.5 Ki 5
MCLMDSQSSOOSRY 9.5 Ki 3
NIPWDBCEPCGPGH 9.5 Ki 3
NIRVMUZGMXCWKU 9.5 Ki 2
XUJMJGTVTZESCM 9.5 Ki 7
XXAHGANHKMWQKV 9.5 Ki 3
YMMRGIIZANFGIG 9.5 Ki 6
BKIXSCDBYYIHQI 9.5 Ki 5
YLDRVNNGBACDSD 9.5 Ki 6
QZDWWRKBDPYMIP 9.5 Ki 6
RGDHMJMNRYQXCW 9.5 Ki 6
LSVOXYMZIGSSNB 9.4 Ki 6
OLKUNPKISSHQBO 9.4 Ki 6
IEDCFFRFAIAYGF 9.4 Ki 7
YVPJMZCJVHJOFG 9.4 Ki 7
ZPSBXQBYCQOCEU 9.4 Ki 6
DKSWXNFPYZCJFU 9.4 Ki 6
HEGJYRQUDMITRQ 9.4 Ki 6
2D structure