Target Details
| UniProt AC | P30989 |
|---|---|
| Gene Symbol | NTSR1 |
| Protein Name | Neurotensin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 118
- Clinical molecules 0
- Avg pChEMBL 8.22
KEGG Pathways (2)
Active Molecules (118)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KDAYPBODTWHIKT
|
6.9 | IC50 | 2 | — | |
IDNHSICEMKTUAB
|
6.8 | Ki | 2 | — | |
BDVMLBCUJHKAHY
|
6.8 | Ki | 2 | — | |
GMRVYKXHXXRDKN
|
6.8 | Ki | 2 | — | |
VAWMSFOVHRCJAX
|
6.7 | Ki | 5 | — | |
FAQZXZDZZXERSD
|
6.7 | Ki | 2 | — | |
PCBPTHDFBQRYJN
|
6.7 | Ki | 2 | — | |
DQDBCHHEIKQPJD
|
6.7 | Ki | 2 | — | |
WCUGKDCOWNIUIM
|
6.7 | Ki | 2 | — | |
JXXKKBSAIYYKNT
|
6.6 | IC50 | 2 | — | |
QPKCTXNJUWXWOS
|
6.6 | Ki | 2 | — | |
SFVVNSFJBCCOAB
|
6.6 | Ki | 2 | — | |
LTVAGLBMDPWQGE
|
6.3 | Ki | 2 | — | |
VUGSOGJXDGZLQH
|
6.3 | Ki | 2 | — | |
MBPNCQJILYQPQH
|
6.2 | Ki | 2 | — | |
SNDVFAKLFRYOKC
|
6.1 | Ki | 2 | — | |
DQDBCHHEIKQPJD
|
6.0 | Ki | 2 | — | |
WCUGKDCOWNIUIM
|
6.0 | Ki | 2 | — |