Target Details
UniProt ACP30989
Gene SymbolNTSR1
Protein NameNeurotensin receptor type 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 118
  • Clinical molecules 0
  • Avg pChEMBL 8.22
Top Co-occurrence Targets
Active Molecules (118)
InChIKey pChEMBL Type Targets Clinical
HMLFJQHLNZZDCB 10.7 IC50 2
CWRXKXKKNUGPMX 9.6 Ki 2
VKGJDQSMFSHQMF 9.6 Ki 2
LLPHZQDUSXFIAY 9.6 IC50 3
UAYFECMCWKVDNR 9.6 Ki 2
UMMPGLLERRQETK 9.6 Ki 2
JQOMFKZSHXBCPP 9.6 IC50 3
KYIGOCCCBXRHNJ 9.6 IC50 43
OTFZHUWITMKDIT 9.6 IC50 3
CFEQRHAHQABPPS 9.5 IC50 3
LNZZSNMCNGPDHL 9.5 IC50 3
MPEPKWMFQGIXEZ 9.5 IC50 3
WCUGKDCOWNIUIM 9.5 Ki 3
JDVIBJLNEIKOTF 9.5 IC50 2
LVYZUBJXPNPGQM 9.5 IC50 2
UTFVODGFXAOPNQ 9.5 IC50 2
TUHCUJKBZKVCAN 9.4 IC50 3
OKIJEOJBCCXHLH 9.4 IC50 2
FDBIFJGWCWHUPD 9.4 IC50 2
KOGXZVUCFKIDJW 9.4 IC50 2
PIFPEOIFYCDCNA 9.4 IC50 3
XRXDWBSFVXUHKZ 9.4 IC50 2
DQDBCHHEIKQPJD 9.4 Ki 2
MAEMKRFOORLALZ 9.4 Ki 5
OVWABJJHOAGNSE 9.3 IC50 3
PCJGZPGTCUMMOT 9.3 IC50 3
WJBXIMDDWCOIEN 9.3 IC50 3
VVYPBQSXUOQLOK 9.3 IC50 3
VXHBEXCNGBFYIK 9.2 IC50 2
DQDBCHHEIKQPJD 9.2 Ki 2
WCUGKDCOWNIUIM 9.2 Ki 2
DQDBCHHEIKQPJD 9.2 Kd 3
WNFLQFAPYRIZST 9.2 Ki 2
YSDMCVFFBDNGNG 9.2 Ki 2
CQDUQLAFKFLQTQ 9.1 Ki 5
BTGHVQLCWVPIKL 9.0 Ki 2
YAKLGSFYTUQYBF 8.9 IC50 3
MNPDUJGZIRLSLW 8.8 IC50 2
XJVLRYYYMKPGCM 8.8 Ki 2
MGSQSJIDCGRMBG 8.7 Ki 2
LJDKIRQGXSOPEQ 8.7 Ki 2
MMHHIRBOAQJREB 8.7 Ki 2
PTMFVPFXWDUXJR 8.6 Ki 5
XDMAKXFFNWEQHI 8.6 Ki 2
LWULHXVBLMWCHO 8.6 IC50 3
ACFFVPRDWLCNQO 8.6 Ki 2
NMKSVHQYWOXLDQ 8.6 Ki 2
WWHHYSHZJPBANK 8.6 Kd 2
PKKAXLATBVZIML 8.6 Ki 2
YUKIPFYNBXVVHA 8.6 Ki 2
2D structure