Target Details
| UniProt AC | P30968 |
|---|---|
| Gene Symbol | GNRHR |
| Protein Name | Gonadotropin-releasing hormone receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 29
- Clinical molecules 0
- Avg pChEMBL 8.21
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AEOBYHAZFRJFPZ
|
9.3 | Ki | 2 | — | |
JZIURJIEJBKSKI
|
9.2 | Ki | 2 | — | |
QNQXCVVLHUSXOW
|
9.1 | IC50 | 2 | — | |
GRKSCYLPVRPFEA
|
9.1 | Ki | 2 | — | |
XGDYFBGSSSIIDK
|
9.1 | IC50 | 2 | — | |
IGTBNUVMBDYPQG
|
8.9 | IC50 | 8 | — | |
QNIZBEIHYCQTEQ
|
8.9 | Ki | 2 | — | |
ZURGVSINFPSAAI
|
8.9 | IC50 | 2 | — | |
WXUZGCQTOVWUDO
|
8.9 | Ki | 2 | — | |
CJUWBZDJMYYRDG
|
8.8 | IC50 | 2 | — | |
YJBAGQATRBRFBC
|
8.8 | IC50 | 2 | — | |
RMVSZBRIILAXIH
|
8.6 | IC50 | 2 | — | |
DOYPVXXUUVHXLK
|
8.5 | Ki | 2 | — | |
FRLGCDYZXBVROR
|
8.4 | Ki | 2 | — | |
MNTVJSYTLLQKAC
|
8.3 | IC50 | 2 | — | |
YGPMVMMFWAZDOJ
|
8.3 | IC50 | 2 | — | |
LHWQBUMJKGGLOH
|
8.3 | Ki | 2 | — | |
HYFHKEYEUYHQDQ
|
8.2 | Ki | 2 | — | |
AVWXVFNJXMOFEK
|
8.1 | Ki | 2 | — | |
KCCHSZZXJXIDAP
|
8.0 | Ki | 2 | — | |
AVEVJMZJJJDOCI
|
7.7 | IC50 | 7 | — | |
PZGSYNNVPNLHQG
|
7.7 | IC50 | 2 | — | |
FDMBTLJSOVSBHD
|
7.5 | Ki | 2 | — | |
ZOMSEVOHXDVESY
|
7.2 | Ki | 2 | — | |
OEBZYYGQPIDGKZ
|
7.2 | Ki | 2 | — | |
SYBXHLIANYBTCO
|
7.1 | Ki | 2 | — | |
CGMLBVPTUVDZPK
|
7.0 | Ki | 2 | — | |
MUIOMNHOLFGIGK
|
6.8 | IC50 | 2 | — | |
ZPFVOMYXTKCCLP
|
6.1 | IC50 | 2 | — |