Target Details
| UniProt AC | P30926 |
|---|---|
| Gene Symbol | CHRNB4 |
| Protein Name | Neuronal acetylcholine receptor subunit beta-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 431
- Clinical molecules 0
- Avg pChEMBL 7.35
KEGG Pathways (4)
Active Molecules (431)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KNSUADXKFTZSIZ
|
6.1 | IC50 | 2 | — | |
RUEDGHCKLGSDLO
|
6.1 | IC50 | 5 | — | |
UQXDPNPETLYQJZ
|
6.1 | Ki | 3 | — | |
VNRFZHXTMQEXQW
|
6.1 | IC50 | 4 | — | |
WXWGOVLEWUNKCM
|
6.1 | IC50 | 5 | — | |
HYDLTSOVXCUHPA
|
6.1 | Ki | 5 | — | |
IJGXBJUJDSODSN
|
6.1 | Ki | 4 | — | |
WJSJLTQPBJXQOW
|
6.1 | Ki | 4 | — | |
ACHWGHFEAPJMKT
|
6.1 | Ki | 5 | — | |
JIGWWGDIEUWCOR
|
6.1 | Ki | 5 | — | |
WJSJLTQPBJXQOW
|
6.1 | Ki | 4 | — | |
XFBDKMSGGGCNAI
|
6.1 | IC50 | 11 | — | |
AWGHJHAVKVZJIW
|
6.1 | Ki | 3 | — | |
MSSOVRDYPAQUAD
|
6.1 | Ki | 3 | — | |
YNFPARFPWZWYJX
|
6.1 | Ki | 2 | — | |
SCQZRFDFSKEVKQ
|
6.0 | Ki | 4 | — | |
WAQCQCZXLRJXOS
|
6.0 | IC50 | 5 | — | |
BKRDDYIAVADMIJ
|
6.0 | Ki | 5 | — | |
DKXYJACKNZCEOQ
|
6.0 | Ki | 3 | — | |
HPYRFABEGFYNNH
|
6.0 | Ki | 2 | — | |
HQDLJJQZMYAAPU
|
6.0 | IC50 | 2 | — | |
ZHZQMBCYDKNEHH
|
6.0 | Ki | 2 | — | |
KKVSVXVHHIOCHW
|
6.0 | Ki | 4 | — | |
KXAAIPFSUGPVMQ
|
6.0 | Ki | 5 | — | |
XNZHLLAIQAZMMY
|
6.0 | IC50 | 4 | — | |
XOEJXZGEXAMGIL
|
6.0 | Ki | 4 | — | |
AGNZBWKVIGAWTQ
|
6.0 | Ki | 3 | — | |
BSAYMXGAHRLDCA
|
6.0 | IC50 | 2 | — | |
DSYBZSDKMVLLBG
|
6.0 | Ki | 3 | — | |
KMIROODCYQMZLK
|
6.0 | Ki | 4 | — | |
NBYYGODJBZAJJF
|
6.0 | IC50 | 2 | — |