Target Details
UniProt ACP30926
Gene SymbolCHRNB4
Protein NameNeuronal acetylcholine receptor subunit beta-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 431
  • Clinical molecules 0
  • Avg pChEMBL 7.35
Top Co-occurrence Targets
Active Molecules (431)
InChIKey pChEMBL Type Targets Clinical
ABPSWEJOHYDZDP 8.8 IC50 11
PGTPXIBBHIHMQS 8.7 IC50 10
PREYWAJYVTVVPE 8.7 IC50 10
GTVWKLSULFFQST 8.7 Ki 7
HGIKFFRIFIJEOP 8.7 IC50 3
WXTQMACZCSXJTB 8.7 Ki 4
PLUODXWJLHWDCV 8.7 Ki 2
NBSDOPKWFMNCQW 8.7 Ki 2
PEYVELBXXMIVMU 8.7 Ki 2
SGVSOCSOUHHZAS 8.7 IC50 3
UIRMNVOEQMAKFM 8.7 IC50 7
MXJPOFBPCRQRTD 8.7 IC50 3
TZWVPYLQJDFQHL 8.7 Ki 5
SLZOZHRDAPBUAU 8.6 IC50 2
ISACHQOCISQFPP 8.6 Ki 4
ZRCMYKLGYHVJGO 8.6 Ki 5
NYPLKEHGCMPSAD 8.6 Ki 2
SWPVFHZSTTYORI 8.6 IC50 5
YSSBTWFASLVAGY 8.6 IC50 5
GLNHQLYIFATJOO 8.6 IC50 3
YRTJBUGCGGXTRV 8.6 IC50 5
HVTMEGQWQQUDIH 8.5 IC50 3
PUMYSIXHQPYXGX 8.5 Ki 4
AGNZBWKVIGAWTQ 8.5 Ki 5
ZRCMYKLGYHVJGO 8.5 Ki 5
COKJMTQIZQACLZ 8.4 IC50 3
OUHSMVDDOPDHGW 8.4 Ki 2
RCSZDVCUNQPLHO 8.4 Ki 7
GIDJZDYNVHMFAH 8.4 IC50 9
QYLKSFXBRALDIS 8.4 IC50 9
BJLKZFUZNNATGZ 8.4 IC50 7
WWXZQSSSEUIZDN 8.3 Ki 2
LYGZRGMHPFAAMR 8.3 Ki 7
ZVMQAHYHODITTD 8.3 Ki 2
NTFKOQBZSNCLLA 8.3 Ki 4
MOMRLMDRIJFWPM 8.3 IC50 5
YDGOUEKZXBLUDG 8.3 IC50 8
TZWVPYLQJDFQHL 8.3 Ki 5
ZLLCEWCZDFPICU 8.3 Ki 5
HQBAWNLKYLZICH 8.2 IC50 3
ATDHPNPDBDEQAK 8.2 IC50 5
BMWDQBTXNBGORC 8.2 IC50 8
GTMXEEZPDPKGRK 8.2 Ki 2
QCSSDCOJCQOKNU 8.2 Ki 5
IELBAACIVCODPI 8.2 IC50 8
QGPJNUIJAGMDMT 8.2 Ki 5
VJEPFPRUUZASOL 8.2 Ki 5
DGQVZUDAKWRJPY 8.2 IC50 8
VVDRDHLUVVGURR 8.2 IC50 5
IMWUFTIDVKJBTJ 8.2 Ki 5
2D structure