Target Details
| UniProt AC | P30876 |
|---|---|
| Gene Symbol | POLR2B |
| Protein Name | DNA-directed RNA polymerase II subunit RPB2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04563 (RNA_pol_Rpb2_1) PF04561 (RNA_pol_Rpb2_2) PF04565 (RNA_pol_Rpb2_3) PF04566 (RNA_pol_Rpb2_4) PF04567 (RNA_pol_Rpb2_5) PF00562 (RNA_pol_Rpb2_6) PF04560 (RNA_pol_Rpb2_7) |
Summary
- Multi-target molecules 2
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (3)
Active Molecules (2)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AAAQFGUYHFJNHI
|
6.9 | IC50 | 252 | — | |
MWKSRKSEWLRPBL
|
6.7 | Kd | 1075 | — |