Target Details
| UniProt AC | P30872 |
|---|---|
| Gene Symbol | SSTR1 |
| Protein Name | Somatostatin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 446
- Clinical molecules 0
- Avg pChEMBL 6.94
KEGG Pathways (4)
Active Molecules (446)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XOPQWKKOVYFZNR
|
8.4 | IC50 | 5 | — | |
ZBJAXLDEWVZEPY
|
8.4 | IC50 | 5 | — | |
MNSYRBDGAPVGIW
|
8.4 | Ki | 4 | — | |
YNCDBNIRPHKYAI
|
8.4 | Ki | 5 | — | |
PPMRXEMNCQTEFU
|
8.4 | IC50 | 5 | — | |
HTEPNQQGQXAYEW
|
8.3 | Ki | 5 | — | |
USUTWRILASMBKB
|
8.3 | IC50 | 3 | — | |
HRXRBQBXRUWBLT
|
8.3 | IC50 | 3 | — | |
ANCUAJMQRRZZNC
|
8.3 | IC50 | 5 | — | |
PJRZZHKHLDKTKL
|
8.3 | IC50 | 5 | — | |
PJRZZHKHLDKTKL
|
8.3 | IC50 | 5 | — | |
PJRZZHKHLDKTKL
|
8.3 | IC50 | 5 | — | |
SJBGEHWYHKHGEN
|
8.3 | Ki | 4 | — | |
HUGAAIZUHOUHDU
|
8.3 | IC50 | 5 | — | |
HUGAAIZUHOUHDU
|
8.3 | IC50 | 5 | — | |
NBHZBFZQSHJQHE
|
8.3 | Kd | 3 | — | |
NBAVJBRNJUQNDP
|
8.2 | IC50 | 2 | — | |
UIVAPXWJQYWBBS
|
8.2 | Ki | 4 | — | |
HSROYJCEDSDMSO
|
8.2 | Ki | 4 | — | |
OOTSWNLCQIKZHR
|
8.2 | Ki | 5 | — | |
VMZMNAABQBOLAK
|
8.2 | Ki | 4 | — | |
UCNKQLMKTJDSDK
|
8.2 | IC50 | 5 | — | |
UCNKQLMKTJDSDK
|
8.2 | IC50 | 5 | — | |
VBPXZFRIJRBHGV
|
8.2 | Ki | 6 | — | |
HMTCBXPQKWFOMG
|
8.2 | Ki | 5 | — | |
ZHTQHERQPPHQPE
|
8.2 | IC50 | 3 | — | |
IMSYGYSLWIQMRP
|
8.1 | IC50 | 3 | — | |
KBPQEKWHQJZFGJ
|
8.1 | Ki | 4 | — | |
LURNPSLHCPCRAL
|
8.1 | IC50 | 2 | — | |
NKLVDXHPTVXWQC
|
8.1 | Ki | 6 | — | |
NIVBKEGMFSFLSD
|
8.0 | IC50 | 5 | — | |
QXFDANJFZYVJAG
|
8.0 | Ki | 5 | — | |
SRQXVUQUEBDWHI
|
8.0 | IC50 | 2 | — | |
UCNKQLMKTJDSDK
|
8.0 | IC50 | 5 | — | |
UCNKQLMKTJDSDK
|
8.0 | IC50 | 5 | — | |
FUIWABOFKJDPGP
|
8.0 | Ki | 4 | — | |
LWKOEELVPGZRCE
|
7.9 | IC50 | 5 | — | |
LWKOEELVPGZRCE
|
7.9 | IC50 | 5 | — | |
BISKEDCOTSGVNU
|
7.8 | IC50 | 2 | — | |
DNESPLSADCEOBA
|
7.8 | IC50 | 5 | — | |
PJRZZHKHLDKTKL
|
7.8 | IC50 | 5 | — | |
YCGSZLSXWAEOFI
|
7.8 | IC50 | 3 | — | |
GIGRDXKZXVSPEN
|
7.8 | IC50 | 2 | — | |
QLVKKYGVIQGKCF
|
7.8 | IC50 | 2 | — | |
UKGIKHPFMXOGRF
|
7.8 | IC50 | 2 | — | |
FJRAPOZDHJLSPN
|
7.8 | IC50 | 2 | — | |
HMHZOCNPBRZNJI
|
7.8 | IC50 | 5 | — | |
MGQOSJMBSMGOOM
|
7.8 | IC50 | 2 | — | |
JNMPZUZCPFIJGJ
|
7.7 | Ki | 5 | — | |
UXKXLWHPLWJRQG
|
7.7 | IC50 | 5 | — |