Target Details
| UniProt AC | P30556 |
|---|---|
| Gene Symbol | AGTR1 |
| Protein Name | Type-1 angiotensin II receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 696
- Clinical molecules 1
- Avg pChEMBL 8.2
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Calcium signaling pathway
- Coronavirus disease - COVID-19
- Cortisol synthesis and secretion
- Cushing syndrome
- Diabetic cardiomyopathy
- Hormone signaling
- Neuroactive ligand-receptor interaction
- Pathways in cancer
- Phospholipase D signaling pathway
- Renin secretion
- Renin-angiotensin system
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Associated Diseases (2)
Active Molecules (696)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTDRSCZZEUAAIP
|
8.8 | Kd | 2 | — | |
GTMLBLOJMPJCBD
|
8.8 | IC50 | 2 | — | |
MLGCITBDCGSKQS
|
8.8 | IC50 | 2 | — | |
RJSWYMPJCFDFTK
|
8.8 | Kd | 2 | — | |
ACKLWEGKSRZTAP
|
8.8 | Kd | 2 | — | |
FRKWBPZUTQTJCZ
|
8.8 | IC50 | 2 | — | |
GBXQWPCVQAHRBS
|
8.8 | IC50 | 2 | — | |
GLWABHJKVIXFLE
|
8.8 | Kd | 2 | — | |
MPBMSFMOTXPLEP
|
8.8 | Kd | 2 | — | |
RQGDXPDTZWGCQI
|
8.8 | Kd | 2 | — | |
MLVRTBMOAVMFSH
|
8.8 | Kd | 2 | — | |
VUFFRQVVDOLRNK
|
8.8 | Kd | 2 | — | |
ISVKMWBCEDWCIW
|
8.8 | Kd | 2 | — | |
JESVDDKOXLZVBB
|
8.8 | IC50 | 2 | — | |
RXKTYMCGYUSQFW
|
8.8 | Kd | 2 | — | |
HQYHXZJKRHOYFK
|
8.7 | IC50 | 2 | — | |
AVAOZIOTPYKTPP
|
8.7 | Kd | 2 | — | |
DDCUEFRQMQCTOM
|
8.7 | IC50 | 2 | — | |
PCJLKHNHECWWOF
|
8.7 | IC50 | 2 | — | |
AAIHSHZCQFBIQU
|
8.7 | IC50 | 2 | — | |
AQTVBIULRJMSFA
|
8.7 | IC50 | 2 | — | |
AXWUCCRVXUGJIS
|
8.7 | IC50 | 2 | — | |
FURKQPPGTMILKC
|
8.7 | IC50 | 2 | — | |
GUILESAVAVIDIH
|
8.7 | IC50 | 2 | — | |
HJBMREOPAOXTDB
|
8.7 | Kd | 2 | — | |
HJWOJDFDUUAQRE
|
8.7 | IC50 | 2 | — | |
HZRZZXFVGPKWLK
|
8.7 | Kd | 2 | — | |
IJRCAHZGYYDUON
|
8.7 | IC50 | 2 | — | |
IYWDGVNLLWLWKC
|
8.7 | IC50 | 2 | — | |
JPWZETSNZSSAFU
|
8.7 | Kd | 2 | — | |
KLLKQECWOKQXKL
|
8.7 | Kd | 2 | — | |
LAUYLCNTECMFDS
|
8.7 | IC50 | 2 | — | |
LPIXEUUSKNZULE
|
8.7 | IC50 | 2 | — | |
MNRJNBDYGPNZPG
|
8.7 | Kd | 2 | — | |
MXXUSTMMIFYSEU
|
8.7 | IC50 | 2 | — | |
NZQIEKNCIJICCT
|
8.7 | IC50 | 2 | — | |
OJBDZHJIPQIGAJ
|
8.7 | IC50 | 2 | — | |
OXCBPWVHMRRTNH
|
8.7 | Kd | 2 | — | |
PGFOMEGDVXUBCE
|
8.7 | IC50 | 2 | — | |
QCRFNJRSBJCWOV
|
8.7 | IC50 | 2 | — | |
RHSHLPBWADWWMO
|
8.7 | IC50 | 2 | — | |
SEDHRMXNXHQPIV
|
8.7 | IC50 | 2 | — | |
SSYKWWYPSOVNMP
|
8.7 | IC50 | 2 | — | |
URJBSQINSKCWSD
|
8.7 | IC50 | 2 | — | |
VVGRGSRZVVXEEN
|
8.7 | IC50 | 2 | — | |
VWWMGPCUZVOLLK
|
8.7 | Kd | 2 | — | |
XMENXPSJCPMABE
|
8.7 | IC50 | 2 | — | |
YOSHYTLCDANDAN
|
8.7 | Ki | 2 | — | |
ZWJUNLRWRHFLJR
|
8.7 | IC50 | 2 | — | |
GABMQILPAPONQS
|
8.7 | IC50 | 2 | — |