Target Details
| UniProt AC | P30556 |
|---|---|
| Gene Symbol | AGTR1 |
| Protein Name | Type-1 angiotensin II receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 696
- Clinical molecules 1
- Avg pChEMBL 8.2
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Calcium signaling pathway
- Coronavirus disease - COVID-19
- Cortisol synthesis and secretion
- Cushing syndrome
- Diabetic cardiomyopathy
- Hormone signaling
- Neuroactive ligand-receptor interaction
- Pathways in cancer
- Phospholipase D signaling pathway
- Renin secretion
- Renin-angiotensin system
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Associated Diseases (2)
Active Molecules (696)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LTIBWTGQXRKVOU
|
9.3 | Kd | 2 | — | |
PHPBPOAOXZGRJY
|
9.3 | IC50 | 2 | — | |
QHRSDSAEHHSTJO
|
9.3 | IC50 | 2 | — | |
RQADEKNPQZFEDJ
|
9.3 | IC50 | 2 | — | |
RULSCFPHIGQRQC
|
9.3 | Kd | 2 | — | |
JCIWYBSLBBKTQW
|
9.3 | Kd | 2 | — | |
BFVNEYDCFJNLGN
|
9.3 | IC50 | 3 | — | |
VGAXZADPFSBRSX
|
9.2 | IC50 | 2 | — | |
WYPIMZRCEFEPBN
|
9.2 | IC50 | 2 | — | |
AADDKLKFCNPPIE
|
9.2 | IC50 | 2 | — | |
BBYKQNJKFVTGSO
|
9.2 | IC50 | 2 | — | |
LKUWPBMJUJRUDE
|
9.2 | IC50 | 2 | — | |
QNRHKXJSLWIGRL
|
9.2 | IC50 | 2 | — | |
QZYYWQARICSTEX
|
9.2 | IC50 | 2 | — | |
TUQUNPUEMOPNAX
|
9.2 | IC50 | 2 | — | |
WKLNGIAELVFRKF
|
9.2 | IC50 | 2 | — | |
XLDPYCCVJVFDNB
|
9.2 | IC50 | 2 | — | |
YQXLJCKCRTVBBJ
|
9.2 | IC50 | 2 | — | |
DYYWUYUUDYPWON
|
9.2 | Kd | 2 | — | |
VBBGBAVUHFREAM
|
9.2 | Kd | 2 | — | |
ZVUNAQTWOGAJRE
|
9.2 | IC50 | 2 | — | |
FDFADTZMGVFJIN
|
9.2 | IC50 | 2 | — | |
GZLUZVHIHGZGIG
|
9.2 | IC50 | 2 | — | |
JASVAUNATQDFDG
|
9.2 | IC50 | 2 | — | |
MEIWZVPKRQJOOT
|
9.2 | IC50 | 2 | — | |
UJTSFCRAAJLWKT
|
9.2 | IC50 | 2 | — | |
WXGFWVAZGIOWBV
|
9.2 | IC50 | 2 | — | |
CZGUSIXMZVURDU
|
9.1 | Ki | 2 | — | |
JHSYCEYHQGMVCC
|
9.1 | IC50 | 2 | — | |
ZKRRGXRLWZULSD
|
9.1 | IC50 | 2 | — | |
LOPJXNWIMDWJRO
|
9.1 | IC50 | 2 | — | |
VPKPMOBKGPHPMM
|
9.1 | Kd | 2 | — | |
YTULTWSYNAMEQG
|
9.1 | IC50 | 2 | — | |
FVRHDLWUNGFIOI
|
9.1 | IC50 | 2 | — | |
GVBCDDWHWJXZHB
|
9.1 | IC50 | 2 | — | |
IMCHWZJWTLLCLS
|
9.1 | Ki | 2 | — | |
LPJUWRWABYMZFP
|
9.1 | IC50 | 2 | — | |
QPYYJLXUFWUYHC
|
9.1 | IC50 | 2 | — | |
WRFHGDPIDHPWIQ
|
9.1 | Ki | 2 | — | |
CWWVFQMJNYJQKE
|
9.1 | IC50 | 2 | — | |
JKXFAOAAQSTEDR
|
9.1 | IC50 | 2 | — | |
TVHACRDUPFKWBO
|
9.1 | IC50 | 2 | — | |
YMJWWFSMUSMMFX
|
9.1 | IC50 | 2 | — | |
SQKIRZKSRXMYJC
|
9.1 | Kd | 2 | — | |
ZVAFXUKVSGFEAS
|
9.1 | Kd | 2 | — | |
GQEYIVWYNBRECD
|
9.1 | IC50 | 2 | — | |
BWSMXLWKVGEYTH
|
9.1 | IC50 | 2 | — | |
YXTFWWJTCDDZKP
|
9.1 | IC50 | 2 | — | |
YZRHNUCZSNUXFT
|
9.1 | IC50 | 2 | — | |
BBGNUQCNZXJBOR
|
9.0 | Kd | 2 | — |