Target Details
| UniProt AC | P30556 |
|---|---|
| Gene Symbol | AGTR1 |
| Protein Name | Type-1 angiotensin II receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 696
- Clinical molecules 1
- Avg pChEMBL 8.2
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Calcium signaling pathway
- Coronavirus disease - COVID-19
- Cortisol synthesis and secretion
- Cushing syndrome
- Diabetic cardiomyopathy
- Hormone signaling
- Neuroactive ligand-receptor interaction
- Pathways in cancer
- Phospholipase D signaling pathway
- Renin secretion
- Renin-angiotensin system
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Associated Diseases (2)
Active Molecules (696)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AAZOKMBAJGOCHB
|
10.9 | Kd | 2 | — | |
DLMNZGAILMQDHA
|
10.4 | Kd | 2 | — | |
OHLFRZINSRPHFC
|
10.3 | Kd | 2 | — | |
YDAHPXSXJZMUPN
|
10.3 | IC50 | 2 | — | |
DANORXBBWTVCPC
|
10.2 | Kd | 2 | — | |
VDFOBEUYPXRSDL
|
10.1 | IC50 | 2 | — | |
KCTFTBCZZUBAKN
|
10.0 | Kd | 2 | — | |
FVTLWMVHJCFCJX
|
10.0 | IC50 | 2 | — | |
HEMRWRORJFHTRV
|
10.0 | IC50 | 2 | — | |
IBRQDSKNQMZKID
|
10.0 | IC50 | 2 | — | |
KBTWUZYANYSHQE
|
10.0 | IC50 | 2 | — | |
NTVPMPFYEITAQZ
|
10.0 | IC50 | 2 | — | |
ODRDBMOWIAECPK
|
10.0 | IC50 | 2 | — | |
PWVCJTQDCHXRDQ
|
10.0 | IC50 | 2 | — | |
QKNPCCKKMYTRGV
|
10.0 | IC50 | 2 | — | |
SLVFZAJWNXKXPD
|
10.0 | IC50 | 2 | — | |
XSVYVIWXYIVSOW
|
10.0 | IC50 | 2 | — | |
XTWVUFDZLCSCDX
|
10.0 | IC50 | 2 | — | |
XZITYYOPLBOABQ
|
10.0 | IC50 | 2 | — | |
XUPVSGKRAWKIFA
|
9.8 | IC50 | 2 | — | |
CFMUZUVRPWGTOR
|
9.8 | IC50 | 2 | — | |
KOGDEEKMGBZZPT
|
9.8 | Kd | 2 | — | |
MHLMVIIDOZELAA
|
9.8 | Kd | 2 | — | |
QRUOLIOKJCMLBE
|
9.8 | Kd | 2 | — | |
ATVZZAXDSVBSGX
|
9.7 | IC50 | 2 | — | |
BELHLEZQMOGSQN
|
9.7 | IC50 | 2 | — | |
CQVJTTOZTTVVBK
|
9.7 | IC50 | 2 | — | |
FNOSMWSPVAMRRG
|
9.7 | IC50 | 2 | — | |
GRVMFLLSNYIYPD
|
9.7 | IC50 | 2 | — | |
LIUNMFCWFYFUGQ
|
9.7 | IC50 | 2 | — | |
LPVSOTPUVUUDBE
|
9.7 | IC50 | 2 | — | |
PBNKWFOVOSXATB
|
9.7 | IC50 | 2 | — | |
PPDJSGSLQZISIW
|
9.7 | IC50 | 2 | — | |
PXHKMVBVVIIYHP
|
9.7 | IC50 | 2 | — | |
QLMPKYMPDFHNLL
|
9.7 | IC50 | 2 | — | |
SGKFZODOLUDBTL
|
9.7 | IC50 | 2 | — | |
SPUPGKSCQBKDNS
|
9.7 | IC50 | 2 | — | |
UHYDTDXHNHZWIN
|
9.7 | IC50 | 2 | — | |
VBGUWLWEBXRIFX
|
9.7 | Kd | 2 | — | |
VVZWXCIUTYOBOD
|
9.7 | IC50 | 2 | — | |
XZXZTTWHUVBVBC
|
9.7 | IC50 | 2 | — | |
ZJAVHMSXOMUSMC
|
9.7 | Kd | 2 | — | |
CRXQSKPJSRFBDS
|
9.7 | Kd | 2 | — | |
QLYHVKQIKYGJHI
|
9.7 | Kd | 2 | — | |
QQMNYPQIZBQLSK
|
9.7 | IC50 | 2 | — | |
ARZUEYHMVSFSTN
|
9.7 | Kd | 2 | — | |
OOEJDMPSOGBATM
|
9.7 | Kd | 2 | — | |
CYNYOKRAMQHBKF
|
9.6 | Kd | 2 | — | |
ISQDDSYNICWABK
|
9.6 | Kd | 2 | — | |
MJFUGUNPGFBNRJ
|
9.6 | Kd | 2 | — |