Target Details
| UniProt AC | P30550 |
|---|---|
| Gene Symbol | GRPR |
| Protein Name | Gastrin-releasing peptide receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 32
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (2)
Active Molecules (32)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BNEIPTFKHBHJBM
|
10.4 | Ki | 2 | — | |
QXZBMSIDSOZZHK
|
9.8 | Ki | 4 | — | |
WPAOEAXJLCSDBY
|
9.8 | IC50 | 2 | — | |
WPAOEAXJLCSDBY
|
9.8 | IC50 | 2 | — | |
IKKYIPCELZIPRY
|
9.6 | IC50 | 3 | — | |
KQHZZRQJOXXKSD
|
9.3 | IC50 | 2 | — | |
KQHZZRQJOXXKSD
|
9.3 | IC50 | 2 | — | |
CDIMJEGYWSSELL
|
9.2 | Ki | 2 | — | |
HGMWCLNMIBXTTP
|
9.2 | Ki | 2 | — | |
BXSSCSKCOFKPOK
|
9.1 | IC50 | 3 | — | |
XDFRCEDKCPCBTG
|
9.1 | IC50 | 2 | — | |
GMEWMQLWXBFPOI
|
9.0 | Ki | 3 | — | |
FAOPTHGFLLUMQK
|
8.4 | Ki | 2 | — | |
NNFUWNLENRUDHR
|
8.4 | IC50 | 2 | — | |
UGDBOJPMQKHDTD
|
8.2 | Ki | 2 | — | |
XPRDWAMLFOLCLZ
|
8.2 | Ki | 2 | — | |
LJRYMIQLJOWZPO
|
8.1 | Ki | 2 | — | |
AFDXUTWMFMAQJO
|
7.8 | Ki | 2 | — | |
YQVMYZMFAIZTCM
|
7.7 | IC50 | 2 | — | |
DMQGYVMAKLBBJM
|
7.5 | Ki | 2 | — | |
VFVKUZVSXDUHAQ
|
7.5 | Ki | 2 | — | |
AFDFFXDMBHJMEI
|
7.5 | Ki | 2 | — | |
ZOKUSEXKSWRJPJ
|
7.4 | Ki | 2 | — | |
YPFNACALNKVZNK
|
7.2 | Ki | 3 | — | |
RNQDZMJJXVOUFD
|
7.1 | Ki | 2 | — | |
XVFAEENKHJXNNB
|
7.1 | Ki | 2 | — | |
YIVURXAOLPNGNO
|
7.0 | Ki | 2 | — | |
ILJBXVQOPJTFJY
|
6.9 | Ki | 2 | — | |
AMIBSGKPRJXHLH
|
6.8 | Ki | 2 | — | |
WUKCFSLNDDXVRY
|
6.6 | Ki | 2 | — | |
IGGDYDYGUOVJQB
|
6.4 | Ki | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |