Target Details
| UniProt AC | P30536 |
|---|---|
| Gene Symbol | TSPO |
| Protein Name | Translocator protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03073 (TspO_MBR) |
Summary
- Multi-target molecules 29
- Clinical molecules 0
- Avg pChEMBL 6.78
KEGG Pathways (3)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CJCIRTWDYKBVBE
|
8.7 | Ki | 2 | — | |
PUMYFTJOWAJIKF
|
8.6 | Kd | 2 | — | |
HSYRKMNHUANBOW
|
8.1 | IC50 | 2 | — | |
RAVIZVQZGXBOQO
|
8.0 | Ki | 2 | — | |
RAVIZVQZGXBOQO
|
7.8 | Ki | 3 | — | |
MWKSRKSEWLRPBL
|
7.6 | Kd | 1075 | — | |
HPAHZCBKRSEDHH
|
7.3 | Ki | 2 | — | |
ZCCPLJOKGAACRT
|
7.0 | Kd | 599 | — | |
BDYNTWOCTIWVBG
|
7.0 | Ki | 2 | — | |
RSYHJSDOGMSLDH
|
7.0 | Ki | 2 | — | |
PMLCQIVFRJHHRF
|
6.9 | Ki | 2 | — | |
MOTJMGVDPWRKOC
|
6.7 | Ki | 2 | — | |
GHMATVSBVUMZAE
|
6.7 | Ki | 2 | — | |
PKJHTQYCVXDPKU
|
6.7 | Ki | 2 | — | |
NXFFJDQHYLNEJK
|
6.5 | Ki | 6 | — | |
UGZASRPZTFYHQC
|
6.4 | Ki | 2 | — | |
TXTXUJCZFZSISJ
|
6.4 | Ki | 2 | — | |
AFRXCTUPOJKNDG
|
6.3 | Ki | 3 | — | |
GXGVWEMSSIKHOZ
|
6.3 | Ki | 8 | — | |
BJIUKEMXFQJDBZ
|
6.2 | Ki | 2 | — | |
BHIJCDLCYUTQCS
|
6.1 | Ki | 2 | — | |
BPRNMVDTWIHULJ
|
6.1 | Ki | 6 | — | |
HYBZWVLPALMACV
|
6.1 | Ki | 4 | — | |
RDONXGFGWSSFMY
|
6.1 | IC50 | 6 | — | |
PCMHOSYCWRRHTG
|
6.1 | Ki | 3 | — | |
SVJMLYUFVDMUHP
|
6.0 | Ki | 26 | — | |
DSEJCLDJIFTPPH
|
6.0 | Ki | 4 | — | |
JENSDTKXNVHSSN
|
6.0 | Ki | 4 | — | |
VAUKHARIAMDAGF
|
6.0 | Ki | 3 | — |