Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NUTKAHHQRZGHIS
|
7.8 | IC50 | 2 | — | |
HNDZJFGTHKMGAS
|
7.8 | IC50 | 3 | — | |
HZJTYICHFKEZPB
|
7.8 | IC50 | 4 | — | |
LZOJVTCTBSNNNT
|
7.8 | IC50 | 4 | — | |
SCPFYDCGZSWLOY
|
7.8 | IC50 | 4 | — | |
YTXPYXBASKYQMU
|
7.8 | IC50 | 2 | — | |
CKRJSIFFXMHDSE
|
7.8 | IC50 | 3 | Yes | |
PZRVIBIFSSVDAU
|
7.8 | IC50 | 2 | — | |
WCKQZMCXHJVIQF
|
7.8 | IC50 | 2 | — | |
BYEDBMHYWDHELH
|
7.7 | IC50 | 2 | — | |
FXTJCTYAPOCFAC
|
7.7 | IC50 | 4 | — | |
LWRKDFICEDGLMK
|
7.7 | IC50 | 2 | — | |
PCYYUIIBSKPSCD
|
7.7 | IC50 | 2 | — | |
QEWWRQLOXCSNGA
|
7.7 | IC50 | 2 | — | |
IQIVRGUWXKHLHL
|
7.7 | IC50 | 2 | — | |
BQOPPXMDAUTYSM
|
7.7 | IC50 | 2 | — | |
KHCNBZBQEJGAOZ
|
7.7 | IC50 | 2 | — | |
LYXOBSREVZDKST
|
7.7 | IC50 | 9 | — | |
NFLIEDMYXBZROG
|
7.7 | IC50 | 2 | — | |
SLCVMWQKWVHPQE
|
7.7 | IC50 | 3 | — | |
SPERNPFVNHOOND
|
7.7 | IC50 | 2 | — | |
IELXVRGBXDSTMS
|
7.7 | IC50 | 2 | — | |
AREYWCZYVPSHGS
|
7.7 | IC50 | 5 | — | |
DKSNLQYRZJKYOC
|
7.7 | Ki | 51 | — | |
DQMZBEHEUJDCNM
|
7.7 | IC50 | 3 | — | |
GCYXEGSPUDSZJY
|
7.7 | Ki | 82 | — | |
NWAUBAGBGOPJLF
|
7.7 | Ki | 51 | Yes | |
XBYVOPRDASFDMY
|
7.7 | Ki | 42 | — | |
XHORJSJFHVABEA
|
7.7 | Ki | 49 | — | |
ZWVZORIKUNOTCS
|
7.7 | Ki | 69 | — | |
ADLLAPNUCPCMFE
|
7.7 | IC50 | 2 | — | |
CWRXCQQDEOGGAA
|
7.7 | IC50 | 2 | — | |
DXASYTJLINRTNC
|
7.7 | IC50 | 4 | — | |
GGVWIGDCUUVFSZ
|
7.7 | IC50 | 4 | — | |
IEXXROGGKUBLPS
|
7.7 | IC50 | 4 | — | |
RQMXEHSOMYFNKM
|
7.7 | IC50 | 2 | — | |
YUAALFPUEOYPNX
|
7.7 | IC50 | 3 | — | |
BBEKTQZNBOIUQG
|
7.7 | IC50 | 2 | — | |
DCFNMFYAKVXCLN
|
7.7 | IC50 | 4 | — | |
UKMXSBKKSKVHAG
|
7.7 | IC50 | 2 | — | |
AKCLLMQIJOIPAK
|
7.6 | IC50 | 2 | — | |
ISOYAPPKZDNVQA
|
7.6 | IC50 | 3 | — | |
JNOZPOGAIWIGDX
|
7.6 | IC50 | 3 | — | |
MBDXRRFVBRTNPY
|
7.6 | IC50 | 2 | — | |
OPBXCUWAHPDQBE
|
7.6 | IC50 | 3 | — | |
PTRVZEMPNWFZEI
|
7.6 | IC50 | 4 | — | |
RCQLJPMEVONOSW
|
7.6 | IC50 | 4 | — | |
WDSAJBCCUSPKPI
|
7.6 | IC50 | 2 | — | |
GKFUTHVAVQPTFA
|
7.6 | IC50 | 2 | — | |
GKTJDVXAUIHAML
|
7.6 | IC50 | 4 | — |