Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
7.9 | Kd | 231 | Yes | |
WTCQJADHNRKLTQ
|
7.9 | IC50 | 2 | — | |
WYEUDIXCTGHYOQ
|
7.9 | IC50 | 2 | — | |
XZWGQOPSCIYJJG
|
7.9 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.9 | Kd | 165 | Yes | |
YKSFAELRDYTAHZ
|
7.9 | IC50 | 3 | — | |
GEGCXGMFUYJULA
|
7.9 | Ki | 30 | Yes | |
RWEHAHIEUDLKGT
|
7.9 | Ki | 33 | — | |
ZVWRFVCNQOECJS
|
7.9 | Ki | 71 | — | |
AKWLDQDWZNJYKL
|
7.9 | IC50 | 14 | — | |
HQMSWMADUGUYFF
|
7.9 | IC50 | 4 | — | |
YWILRIPPYUJHMX
|
7.9 | IC50 | 4 | — | |
HXCACITXFCPZQQ
|
7.9 | IC50 | 2 | — | |
KXMZDGSRSGHMMK
|
7.8 | IC50 | 14 | — | |
MJSHVHLADKXCML
|
7.8 | IC50 | 11 | — | |
MJSHVHLADKXCML
|
7.8 | IC50 | 4 | — | |
QORFKFBKAXIHDO
|
7.8 | IC50 | 2 | — | |
SSJIQTZEUSHBBQ
|
7.8 | IC50 | 4 | — | |
TUSFBIZKPNHLKT
|
7.8 | IC50 | 4 | — | |
ULIRDGCRHUZAAA
|
7.8 | IC50 | 2 | — | |
UTPPAOMSIMPNEQ
|
7.8 | IC50 | 4 | — | |
BCOMIOVRJUNIKO
|
7.8 | IC50 | 2 | — | |
LBEJYFVJIPQSNX
|
7.8 | IC50 | 4 | — | |
MCRHIHOQPHSEMM
|
7.8 | IC50 | 2 | — | |
ORRNXRYWGDUDOG
|
7.8 | IC50 | 5 | — | |
RGJASBGADDXMBE
|
7.8 | IC50 | 4 | — | |
YWPWDZZAROUKLO
|
7.8 | IC50 | 2 | — | |
HQVWTQMEFOONTI
|
7.8 | IC50 | 2 | — | |
BIKYDWLMTPRSQL
|
7.8 | Ki | 50 | — | |
BOTRGRDIRVJRGQ
|
7.8 | IC50 | 2 | — | |
DPXCMTQMIGMPBI
|
7.8 | IC50 | 2 | — | |
FPLGAASDZAAKLR
|
7.8 | IC50 | 2 | — | |
GMYYMEOGFRKSFS
|
7.8 | Ki | 29 | — | |
GWMATETWMAQOFL
|
7.8 | Ki | 36 | — | |
HCNIBOQWDVOZKF
|
7.8 | Ki | 26 | — | |
HMFLIEILARDTTE
|
7.8 | IC50 | 2 | — | |
HRZOUBQYVUXBNS
|
7.8 | Ki | 38 | — | |
IBLUITUCVORWLC
|
7.8 | IC50 | 3 | — | |
JXNMCDLXYWQTIW
|
7.8 | Ki | 13 | — | |
LWZKYWNWDTZZGI
|
7.8 | IC50 | 3 | — | |
MHCPAORAYMTGCZ
|
7.8 | Ki | 37 | — | |
PUPCRRRSBUYJAD
|
7.8 | Ki | 44 | Yes | |
RWENGGARDXLTTR
|
7.8 | IC50 | 3 | — | |
SPZDCHRXPBSIHM
|
7.8 | IC50 | 6 | — | |
VTXUNTHLMBMYAD
|
7.8 | IC50 | 2 | — | |
VXENEMCDVCFWGW
|
7.8 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
7.8 | Ki | 66 | — | |
XBBFRFFVOXSJOR
|
7.8 | IC50 | 2 | — | |
XLFYOIVELARSKP
|
7.8 | Ki | 33 | — | |
AJBIYXUNQZYBRC
|
7.8 | IC50 | 3 | — |