Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GUBJNPWVIUFSTR
|
8.1 | IC50 | 103 | — | |
LPVZJEBCLVVMCF
|
8.1 | IC50 | 2 | — | |
MVJMMLFMPWITEJ
|
8.1 | Ki | 110 | — | |
QONPPIZSNSSCSK
|
8.1 | Ki | 45 | Yes | |
XQTQDOHPJHEUPU
|
8.1 | IC50 | 2 | — | |
HTZHPXKKPOLGTR
|
8.1 | IC50 | 9 | — | |
JITFHFSUXWQAPS
|
8.1 | IC50 | 2 | — | |
RVQLPUNPSVMPIU
|
8.1 | IC50 | 2 | — | |
JLUXEIBYLLFPTR
|
8.1 | IC50 | 2 | — | |
ODHHBTQTAVNJQP
|
8.1 | IC50 | 2 | — | |
GPQKRDLDDKHLKK
|
8.1 | IC50 | 2 | — | |
LDYZXHSJFDQENC
|
8.1 | IC50 | 2 | — | |
OSQTZXWCOXMSCA
|
8.1 | IC50 | 2 | — | |
XFDWKMREXUNRTL
|
8.1 | IC50 | 2 | — | |
DGMFNZXEGKFREH
|
8.1 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
8.1 | Kd | 201 | Yes | |
XBVQPBVYQLZBGU
|
8.1 | IC50 | 2 | — | |
HQDFMNJNVUENSH
|
8.0 | IC50 | 2 | — | |
USGGKJZAODNEBP
|
8.0 | IC50 | 2 | — | |
IKQPJOFHAZFMNC
|
8.0 | IC50 | 4 | — | |
ISPBCAXOSOLFME
|
8.0 | IC50 | 11 | — | |
PHYBXPXVBJFNTE
|
8.0 | IC50 | 2 | — | |
MRKQEMFQARHIQR
|
8.0 | IC50 | 2 | — | |
BSFNGHCTZDCQBF
|
8.0 | Ki | 93 | — | |
FWXIWEQAGQKYSB
|
8.0 | IC50 | 4 | — | |
GRUNJVATCGAOIE
|
8.0 | IC50 | 2 | — | |
IRBBFXPKIBQFKT
|
8.0 | IC50 | 5 | — | |
JMSXCJHWSPPQRP
|
8.0 | IC50 | 3 | — | |
LBEJYFVJIPQSNX
|
8.0 | IC50 | 4 | — | |
NCGOROUZONSZHC
|
8.0 | IC50 | 2 | — | |
OWFXKTOLFUQPDJ
|
8.0 | Ki | 36 | — | |
QIRBYYSKWYYQEJ
|
8.0 | IC50 | 3 | — | |
RGAZVGZUBCFHRJ
|
8.0 | IC50 | 5 | — | |
SJQFBBFEPIQMHG
|
8.0 | IC50 | 2 | — | |
YEPNVBNYCRGZRX
|
8.0 | Ki | 26 | — | |
LJTUUVXTQQTMTB
|
8.0 | IC50 | 2 | — | |
XJVOXPBGMZCIJM
|
8.0 | IC50 | 2 | — | |
BPOGHKOSOWZBGZ
|
8.0 | IC50 | 4 | — | |
CXQHYVUVSFXTMY
|
8.0 | IC50 | 154 | — | |
DVJHTWUZFJCMII
|
8.0 | IC50 | 2 | — | |
QHBNTQCVLLJAGG
|
8.0 | IC50 | 4 | — | |
QIJNQRCCSXIKCW
|
8.0 | IC50 | 2 | — | |
QLBFPPCIKGUBAH
|
8.0 | IC50 | 4 | — | |
QOMGQLZYIUPQLG
|
8.0 | IC50 | 7 | — | |
RJTVPQLMBWIFKC
|
8.0 | IC50 | 5 | — | |
UTBNTDYEJRQXQB
|
8.0 | IC50 | 2 | — | |
VQYYQSZNRVQLIS
|
8.0 | IC50 | 3 | — | |
APJOBTGOJXGDGH
|
7.9 | IC50 | 2 | — | |
HWCUOHGOTYDJTF
|
7.9 | IC50 | 2 | — | |
MCPVQJIWQOAKGR
|
7.9 | IC50 | 2 | — |