Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MVPRWLBKNHWFPM
|
8.2 | IC50 | 6 | — | |
UFCSFQQMMHEHHY
|
8.2 | IC50 | 2 | — | |
UGAWJRIPKFUXGB
|
8.2 | IC50 | 2 | — | |
AZIQVRPNDXMEOX
|
8.2 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
8.2 | Ki | 44 | — | |
ATNVOCQRWNYCHO
|
8.2 | IC50 | 2 | — | |
DZSUJUOJJJCWGG
|
8.2 | Ki | 55 | Yes | |
LGHBDVLAHHANMX
|
8.2 | Ki | 53 | — | |
RIWPMLGHVQKIKL
|
8.2 | IC50 | 2 | — | |
WUPLDKYYIOASBT
|
8.2 | IC50 | 2 | — | |
XKZINYYXWJEYEL
|
8.2 | Ki | 37 | — | |
DXPSQKSTVIVZLV
|
8.2 | IC50 | 6 | Yes | |
AWOJPBWFDKHWTR
|
8.2 | IC50 | 2 | — | |
VUWNSIKRZRWGIE
|
8.2 | IC50 | 2 | — | |
VVQFSZLHAOOPPI
|
8.2 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.2 | Kd | 213 | — | |
PRHOXIYUALUHTC
|
8.2 | IC50 | 2 | — | |
URJHRMXSWREGLT
|
8.2 | IC50 | 2 | — | |
XRLWMHNBPLXCKL
|
8.2 | IC50 | 2 | — | |
FKCWHHYUMFGOPY
|
8.2 | IC50 | 2 | — | |
ITGCBNCSACPXID
|
8.2 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
8.2 | Ki | 48 | — | |
MUCGSGOMAYJYJQ
|
8.2 | IC50 | 2 | — | |
NBKAWHPTEZYULQ
|
8.2 | IC50 | 2 | — | |
ONIQOQHATWINJY
|
8.2 | IC50 | 25 | — | |
IQOCOGQTLHXQMU
|
8.1 | IC50 | 2 | — | |
NEAJWUKNRWPSCI
|
8.1 | IC50 | 2 | — | |
RQZDAXOPNDQREW
|
8.1 | IC50 | 2 | — | |
UFBWCXYTJNSQAR
|
8.1 | IC50 | 2 | — | |
MGGANBWHQUWTFD
|
8.1 | IC50 | 3 | — | |
QJRBENOWXGFKIL
|
8.1 | IC50 | 2 | — | |
XIBKNASIQNAJFG
|
8.1 | IC50 | 2 | — | |
BSBDXSGQMHVOLT
|
8.1 | IC50 | 2 | — | |
KQVZUBPWFJXMKN
|
8.1 | IC50 | 3 | — | |
LLGTZIXASKDKRV
|
8.1 | IC50 | 2 | — | |
LMKSUPHSUOCPTM
|
8.1 | IC50 | 2 | — | |
NFCXQIHBUDNOQY
|
8.1 | IC50 | 2 | — | |
NPMHPYDYYNJHLT
|
8.1 | IC50 | 2 | — | |
UKJAACLEQSSYIE
|
8.1 | IC50 | 2 | — | |
VRBCYHMHHGOSNK
|
8.1 | IC50 | 2 | — | |
WDXBRUHVKWGDOP
|
8.1 | IC50 | 2 | — | |
WRADGJQBDXJRIT
|
8.1 | IC50 | 2 | — | |
YOSQZDHYWPCOKE
|
8.1 | IC50 | 2 | — | |
ZMODBJGIKIUPSW
|
8.1 | IC50 | 2 | — | |
ZPBNHZZNPPBHBE
|
8.1 | IC50 | 2 | — | |
ZYCWFLSNKRWWQH
|
8.1 | IC50 | 2 | — | |
YINIQNXRRAYBRJ
|
8.1 | IC50 | 2 | — | |
CFIBXVQLBVNOHW
|
8.1 | Ki | 64 | — | |
GSXRCPJTNIGKSZ
|
8.1 | Ki | 43 | — |