Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEVCBWKJSOLMNQ
|
8.4 | Ki | 38 | — | |
UOOZSMNSBYVUGZ
|
8.4 | Ki | 32 | — | |
YIEKEILDJWQXRB
|
8.4 | IC50 | 4 | — | |
YYFOSKNQHFIIIM
|
8.4 | IC50 | 2 | — | |
PVPLEDXJDAJQPM
|
8.4 | IC50 | 2 | — | |
SLRINRCTDNIRFQ
|
8.4 | IC50 | 3 | — | |
CRJMKZAXSRYICG
|
8.4 | IC50 | 2 | — | |
DKZQQJXYLNUWFT
|
8.4 | IC50 | 4 | — | |
UXHQCLFISGGSLE
|
8.4 | IC50 | 2 | — | |
JXOOCVOCZKLKCJ
|
8.4 | IC50 | 2 | — | |
PRISLGCTIWIYSJ
|
8.4 | IC50 | 2 | — | |
WPBQHEXHVOGJHS
|
8.4 | IC50 | 2 | — | |
BZXGAOVHQLAFCU
|
8.4 | IC50 | 2 | — | |
OBTYAQOWQNEKBT
|
8.4 | IC50 | 2 | — | |
SZWMZMVQRXLMGH
|
8.4 | IC50 | 2 | — | |
UOUHQYNDRQLKBR
|
8.4 | IC50 | 2 | — | |
XDXHFPNTAVKXEG
|
8.4 | IC50 | 2 | — | |
XWIZWSBWIAVPBR
|
8.4 | IC50 | 3 | — | |
MFZSNXAYRLASRN
|
8.3 | IC50 | 2 | — | |
MBSLAWMYDOHYMD
|
8.3 | IC50 | 2 | — | |
UIGHJEVAFXUSJH
|
8.3 | IC50 | 2 | — | |
BEDLWZIQKBYUTB
|
8.3 | IC50 | 2 | — | |
GGSXJCQIMZWBFQ
|
8.3 | IC50 | 2 | — | |
YCGFHHACUCVQPI
|
8.3 | IC50 | 2 | — | |
YRANDDHDKOLWES
|
8.3 | IC50 | 2 | — | |
GHZOFMBOCOPIGL
|
8.3 | IC50 | 2 | — | |
HNAKLVMXRNMVMX
|
8.3 | IC50 | 2 | — | |
AMOJZZNHYLYYBD
|
8.3 | IC50 | 2 | — | |
HPBXBZWZAPICIM
|
8.3 | IC50 | 2 | — | |
JNVFMMAYSXTMTJ
|
8.3 | IC50 | 2 | — | |
MPWQARZLUHZHMX
|
8.3 | IC50 | 2 | — | |
NRGYZNJPCGRCLV
|
8.3 | Ki | 52 | — | |
WWFWWACWIOTPBI
|
8.3 | IC50 | 2 | — | |
MWCJYALAMCYPDD
|
8.3 | IC50 | 2 | — | |
YLSAFDQGYSUAFT
|
8.3 | IC50 | 2 | — | |
JRFAYFIOQCIYFZ
|
8.3 | IC50 | 2 | — | |
SAIJSXPUPZBTMI
|
8.3 | IC50 | 2 | — | |
UBJLGYQQFARAFL
|
8.3 | IC50 | 2 | — | |
UEMPFKOYBHCUIG
|
8.3 | IC50 | 4 | — | |
YLKNZRZBRWCKRM
|
8.3 | IC50 | 2 | — | |
JKQBDGDSVVQSGS
|
8.3 | IC50 | 2 | — | |
UGAWJRIPKFUXGB
|
8.3 | IC50 | 2 | — | |
GKKZRQXWOXFPPU
|
8.3 | IC50 | 2 | — | |
XUZJQPLUDYDVEN
|
8.3 | IC50 | 2 | — | |
CXQUSKUCZSYVLJ
|
8.2 | IC50 | 2 | — | |
DRBYDXGARLXEMD
|
8.2 | IC50 | 2 | — | |
RYQKZEFCGLDZCP
|
8.2 | IC50 | 2 | — | |
XSIQDWROCVFQSV
|
8.2 | IC50 | 2 | — | |
COSVDEYENWRMCL
|
8.2 | IC50 | 3 | — | |
LJCANGDUIWZUBX
|
8.2 | IC50 | 2 | — |