Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMXFKJMRDGGNKM
|
8.5 | IC50 | 3 | — | |
ZHHWIWQMTHPAOR
|
8.5 | IC50 | 2 | — | |
IEJMTNVTRDPUHP
|
8.5 | IC50 | 2 | — | |
MYRCTKCEUUSBDZ
|
8.5 | IC50 | 2 | — | |
OYFAPWKIKGMNQO
|
8.5 | IC50 | 2 | — | |
YLSAFDQGYSUAFT
|
8.5 | IC50 | 2 | — | |
YUKVQCUADDDWFR
|
8.5 | IC50 | 2 | — | |
HLKNAIHDOGWCMT
|
8.5 | IC50 | 2 | — | |
IITRYWKRMYPEEH
|
8.5 | IC50 | 2 | — | |
LGWOKPLTMXFKLZ
|
8.5 | IC50 | 2 | — | |
MGETVYBTJTWGJG
|
8.5 | IC50 | 2 | — | |
SLRXPNTXSLSWEL
|
8.5 | IC50 | 2 | — | |
VRDGZPOCAQZKMY
|
8.5 | IC50 | 2 | — | |
WWYZAHWIUVISIK
|
8.5 | IC50 | 2 | — | |
ZMTGUZWATGQQFE
|
8.5 | IC50 | 2 | — | |
DWUNWBPFOCBLPR
|
8.5 | IC50 | 2 | — | |
HKZKELVPGXJIMW
|
8.5 | Ki | 41 | — | |
PYXQMJSGJIJHJT
|
8.5 | Ki | 28 | — | |
SFPWNTQWFFNJIH
|
8.5 | Ki | 48 | — | |
ULMCFLZUGRSEQA
|
8.5 | Ki | 17 | — | |
XYXLUJQBBIBJFV
|
8.5 | Ki | 36 | — | |
RWOFWISHLYBHDE
|
8.5 | IC50 | 2 | — | |
UZXNBLXFPDDYST
|
8.5 | IC50 | 2 | — | |
XSXUZWJPMJGSJV
|
8.5 | IC50 | 2 | — | |
BIOCOIJRRXEMAB
|
8.5 | IC50 | 2 | — | |
GBDADLBKHYUAQL
|
8.5 | IC50 | 2 | — | |
FQIGYFHTRSLGKQ
|
8.5 | IC50 | 2 | — | |
GINRVSOEUKVVID
|
8.5 | IC50 | 2 | — | |
NPPNDOYKLAXXAS
|
8.5 | IC50 | 2 | — | |
ZNVICUGUUAWZQJ
|
8.5 | IC50 | 2 | — | |
OSKAWGHRJOWPNQ
|
8.4 | IC50 | 2 | — | |
YCXZBULDUGDETC
|
8.4 | IC50 | 2 | — | |
DJSUVZWWNNNEDR
|
8.4 | IC50 | 2 | — | |
OZIZRJFBDUUQNT
|
8.4 | IC50 | 3 | — | |
PTQDZIAZJFMTIT
|
8.4 | IC50 | 2 | — | |
AGDRQXKCLKCKEA
|
8.4 | IC50 | 2 | — | |
DAOGGCDCTXWDAX
|
8.4 | IC50 | 2 | — | |
DNXCFFPPWFGXKA
|
8.4 | IC50 | 3 | — | |
GEMNVMUNTRERDJ
|
8.4 | IC50 | 2 | — | |
NBXADWAEHKGGJP
|
8.4 | IC50 | 2 | — | |
WZXCBFSKSWUTOQ
|
8.4 | IC50 | 2 | — | |
GVCDBKPGHJYKCP
|
8.4 | IC50 | 2 | — | |
KYIVMAWNIPIMAX
|
8.4 | IC50 | 2 | — | |
PWNYLFPOEAFAPH
|
8.4 | IC50 | 2 | — | |
VEAHCSCQSILXPX
|
8.4 | IC50 | 2 | — | |
XTKBOFNZDPSRBW
|
8.4 | IC50 | 2 | — | |
IHPWXCGLDDMKCX
|
8.4 | IC50 | 2 | — | |
NSYLBOUGDLOZHC
|
8.4 | IC50 | 2 | — | |
FLMRVDLSUJPCPS
|
8.4 | IC50 | 3 | — | |
KSZDMKRJEQNXAQ
|
8.4 | IC50 | 3 | — |