Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LFNLHBNNYPVNJY
|
8.7 | IC50 | 2 | — | |
QHADVLVFMKEIIP
|
8.7 | IC50 | 9 | — | |
QPIHEOATRHIZAP
|
8.7 | IC50 | 2 | — | |
RBXYGQNZRVPDNB
|
8.7 | Ki | 34 | — | |
RQAATFYANFZYNJ
|
8.7 | IC50 | 2 | — | |
UFGKRFSRVWAORW
|
8.7 | IC50 | 2 | — | |
XOOAAYRIVATZNM
|
8.7 | Ki | 55 | — | |
CYWYLXHLHZXEMX
|
8.7 | IC50 | 2 | — | |
HXGIQMKSZVMZAD
|
8.7 | IC50 | 2 | — | |
PHACAAIWJAWPHA
|
8.7 | IC50 | 2 | — | |
UDHIJSWGTJKLCI
|
8.7 | IC50 | 2 | — | |
SBKRTFFWDDCQLH
|
8.7 | IC50 | 2 | — | |
XCXMZUYZFOFSTB
|
8.7 | IC50 | 2 | — | |
YLKPPBUPVVBPDB
|
8.7 | IC50 | 2 | — | |
FFJXATKZPJXQMA
|
8.7 | IC50 | 2 | — | |
SKYHCUQSFHNVGB
|
8.7 | IC50 | 2 | — | |
IOIMKJTYVDQVKR
|
8.6 | IC50 | 2 | — | |
LZHNGGOUJMOCJB
|
8.6 | IC50 | 2 | — | |
OMLSWMSNQYAKOY
|
8.6 | IC50 | 2 | — | |
VXVHXDKIVTYZHG
|
8.6 | IC50 | 2 | — | |
WPSAGYVBZPKGAO
|
8.6 | IC50 | 2 | — | |
WLTXIECTWSMSQB
|
8.6 | IC50 | 2 | — | |
AQBVKZHNZSNTDM
|
8.6 | IC50 | 2 | — | |
RWHXYPTULXPVSO
|
8.6 | IC50 | 2 | — | |
YQDQJTHWHPDCGQ
|
8.6 | IC50 | 2 | — | |
ZNORSSZINYHFFL
|
8.6 | IC50 | 2 | — | |
ZPWPDCBMIRNATA
|
8.6 | IC50 | 2 | — | |
KBRRUGLLZHVECV
|
8.6 | IC50 | 2 | — | |
MULNSLQVKKUPJN
|
8.6 | Ki | 41 | — | |
WFAOCMRUJDNSOA
|
8.6 | IC50 | 2 | — | |
XVJQKOIBNAWHNV
|
8.6 | IC50 | 2 | — | |
YCGFHHACUCVQPI
|
8.6 | IC50 | 2 | — | |
ZOEILZXFYPPMTR
|
8.6 | IC50 | 2 | — | |
SEXXDGZEFCIZGQ
|
8.6 | IC50 | 2 | — | |
UWVZGNPCAGNKPM
|
8.6 | IC50 | 2 | — | |
WFHGEWDDDBUGKR
|
8.6 | IC50 | 2 | — | |
ZEQSGOFKTMWPAI
|
8.6 | IC50 | 2 | — | |
BHQBNRDVYQVMDL
|
8.6 | IC50 | 2 | — | |
FUKYTTWUNYCSJG
|
8.6 | IC50 | 2 | — | |
HFOSJCQJOTUBNX
|
8.6 | IC50 | 2 | — | |
IKENQUDOTQBCJH
|
8.6 | Kd | 18 | — | |
OVKBEVSXNZKSNI
|
8.6 | IC50 | 2 | — | |
NKPMZIRBMWWISL
|
8.6 | IC50 | 2 | — | |
ZOEILZXFYPPMTR
|
8.6 | IC50 | 2 | — | |
AGPYHKUKKNTOOF
|
8.6 | IC50 | 2 | — | |
QWSBWFZCNLMQCF
|
8.6 | IC50 | 2 | — | |
YJZTUFCHNMWPJK
|
8.6 | IC50 | 2 | — | |
DRUZOODDDHIXAI
|
8.5 | IC50 | 2 | — | |
VJBZMEXUEJVLAU
|
8.5 | IC50 | 2 | — | |
WZIASJJBXMZPDE
|
8.5 | IC50 | 2 | — |