Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OUJHQVBNJZKTSS
|
9.0 | IC50 | 2 | — | |
TZFAMUMVJZGJNK
|
9.0 | IC50 | 2 | — | |
VOMZTXKSRXWVTR
|
9.0 | IC50 | 2 | — | |
XHIQDQUOOKVPRP
|
9.0 | IC50 | 4 | — | |
CQHNWEKZZSCARI
|
8.9 | IC50 | 2 | — | |
GVZMDMVDKHKLPJ
|
8.9 | IC50 | 2 | — | |
JYSXNODIVIMDDT
|
8.9 | IC50 | 2 | — | |
LBFYYFRPBFRKSE
|
8.9 | IC50 | 2 | — | |
LZLIMPWYCRFCKB
|
8.9 | IC50 | 2 | — | |
OQLLSZTVSXCTIX
|
8.9 | IC50 | 2 | — | |
ZIEVFEZSDLFCCS
|
8.9 | IC50 | 2 | — | |
WHMMKPWGWNYYFE
|
8.9 | IC50 | 2 | — | |
MQRDVGBWWVWMEN
|
8.9 | Ki | 47 | — | |
PTVPBWWDGZSEAF
|
8.9 | Ki | 63 | — | |
VKBFHTIUXUCYRQ
|
8.9 | Ki | 66 | — | |
DBAIZGMGQSAOER
|
8.9 | IC50 | 2 | — | |
DVYVSTMPCPXIIT
|
8.9 | IC50 | 2 | — | |
NBWPBWVCXDBJIJ
|
8.9 | IC50 | 2 | — | |
PXNSUHQVXVDKFQ
|
8.9 | IC50 | 2 | — | |
AIIRAHKUAWNOHT
|
8.8 | IC50 | 2 | — | |
ASMANSOISNDQDG
|
8.8 | IC50 | 2 | — | |
FAOUZNFWHWLTIC
|
8.8 | IC50 | 3 | — | |
KIMZAWNVESXXES
|
8.8 | IC50 | 2 | — | |
MYBMVTCYUBVOEK
|
8.8 | IC50 | 2 | — | |
VNBRGSXVFBYQNN
|
8.8 | IC50 | 22 | Yes | |
MQZVKSLKRZNVIE
|
8.8 | IC50 | 2 | — | |
RFBIIBVIVNVJSA
|
8.8 | IC50 | 2 | — | |
UOIRCOJSMABXQO
|
8.8 | IC50 | 2 | — | |
WLAVZAAODLTUSW
|
8.8 | IC50 | 7 | — | |
XJQJAMKWRLSFRE
|
8.8 | IC50 | 2 | — | |
ACJPYAYXMSVFMW
|
8.8 | IC50 | 2 | — | |
LVUPJIBJEABNLA
|
8.8 | IC50 | 2 | — | |
WPHKIQPVPYJNAX
|
8.8 | Ki | 81 | — | |
YQGUQZWOHCDPTK
|
8.8 | IC50 | 2 | — | |
JVFSAMBNAXDBQY
|
8.8 | IC50 | 2 | — | |
RVDBTAAWJRHFHM
|
8.8 | IC50 | 2 | — | |
MBJBZECMDXNZSX
|
8.8 | IC50 | 2 | — | |
ZOEILZXFYPPMTR
|
8.8 | IC50 | 2 | — | |
AHTUGEFRTOJHHF
|
8.7 | IC50 | 2 | — | |
AUUMOHGHBVZXHF
|
8.7 | IC50 | 2 | — | |
HOXZXBFXGVZLRF
|
8.7 | IC50 | 2 | — | |
LGFIHCKPCBQABH
|
8.7 | IC50 | 2 | — | |
MVHPGOCNSYOLJS
|
8.7 | IC50 | 2 | — | |
PKCOJEQPEFFMMK
|
8.7 | IC50 | 2 | — | |
AEGRAVKQKLWNSA
|
8.7 | IC50 | 2 | — | |
GAYKTWZLTBSKSY
|
8.7 | IC50 | 2 | — | |
HJCZOBLYJWGMDD
|
8.7 | IC50 | 2 | — | |
JXIOZYRODOOPLU
|
8.7 | IC50 | 2 | — | |
LAPPKEKKVUXSCR
|
8.7 | IC50 | 2 | — | |
ATIWZLMXSXMEDE
|
8.7 | IC50 | 2 | — |