Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WERQRDFKILOXSK
|
7.4 | IC50 | 3 | — | |
YLAIGAIPEXSTTK
|
7.4 | IC50 | 3 | — | |
DNINGYYWXPRQDJ
|
7.4 | Kd | 4 | — | |
YBWYETJWZZCBAO
|
7.4 | IC50 | 2 | — | |
CQBBMNXXVMOFCA
|
7.4 | Ki | 39 | — | |
FLEAYYMORDPWAJ
|
7.4 | Ki | 90 | — | |
HAYYBYPASCDWEQ
|
7.4 | Ki | 47 | — | |
HYUGTGGDEAGXJP
|
7.4 | IC50 | 11 | — | |
OYUDNKFIGXAIRZ
|
7.4 | Ki | 16 | Yes | |
PCQMERRARZKTPW
|
7.4 | Ki | 68 | — | |
QKPLUKMJEKRAJD
|
7.4 | Ki | 30 | Yes | |
SMIXLVLRWCBPBA
|
7.4 | IC50 | 4 | — | |
WFTZMAAMCVPJJT
|
7.4 | Ki | 26 | — | |
WUWDLXZGHZSWQZ
|
7.4 | Ki | 41 | — | |
GFETUQKKOOEAQJ
|
7.4 | IC50 | 2 | — | |
LVLFSSZNAIKYCD
|
7.4 | IC50 | 19 | — | |
QJLMOARFSPIREY
|
7.4 | IC50 | 3 | — | |
YULMPWFRJYANBE
|
7.4 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
7.4 | IC50 | 92 | — | |
ZFBBKOBKYNRTOS
|
7.4 | IC50 | 4 | — | |
GDKUSUOIODZPAK
|
7.4 | IC50 | 3 | — | |
NBIOGGWEVWYBFI
|
7.4 | IC50 | 4 | — | |
DCSJNPUSJYLHBA
|
7.4 | IC50 | 3 | — | |
NDWOEUVAOGUXGP
|
7.4 | IC50 | 4 | — | |
YHVAWTSFRPAMNQ
|
7.4 | IC50 | 2 | — | |
ZICDFYRPBWSYAQ
|
7.3 | IC50 | 5 | — | |
JZBDNDJNPAVSSE
|
7.3 | IC50 | 3 | — | |
RCQLJPMEVONOSW
|
7.3 | IC50 | 4 | — | |
WGGIKOGLKDIBTL
|
7.3 | IC50 | 2 | — | |
KVUCOURZIKDXHZ
|
7.3 | IC50 | 4 | — | |
ACNCCUVYXQGPKZ
|
7.3 | Ki | 31 | — | |
IAKGNUWZPSPEKU
|
7.3 | Ki | 19 | — | |
LCGSWTFWYNYUKS
|
7.3 | Ki | 26 | — | |
ORJFNGOUYHBFPE
|
7.3 | IC50 | 4 | — | |
RJZDECGDCKOHBV
|
7.3 | Ki | 70 | — | |
UOYIIWVJEPEEOF
|
7.3 | IC50 | 3 | — | |
UWDBNTXEKYRMSG
|
7.3 | Ki | 26 | — | |
HBQLAXMLLMAJCM
|
7.3 | IC50 | 4 | — | |
NQSLOMAYSOUYFR
|
7.3 | IC50 | 3 | — | |
FSWNWXIANJUKSD
|
7.3 | IC50 | 2 | — | |
GZVQZLVAKXRTHU
|
7.3 | IC50 | 7 | — | |
YVBZLUKOBVRLDZ
|
7.3 | IC50 | 2 | — | |
ADCDBRPCQQHZQR
|
7.3 | IC50 | 2 | — | |
AEDKPHMRPYJLGA
|
7.3 | IC50 | 2 | — | |
AEQQTRGTUZUWBY
|
7.3 | IC50 | 2 | — | |
AGGJFPXHGOZHPV
|
7.3 | IC50 | 2 | — | |
AHWSJOBFFQBHOW
|
7.3 | IC50 | 2 | — | |
ALNVGNKIGFPGCV
|
7.3 | IC50 | 3 | — | |
ANINHDBXZARAPZ
|
7.3 | IC50 | 2 | — | |
ANMIEKMLZVVUCN
|
7.3 | IC50 | 2 | — |