Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SKWKMYGZRULQCM
|
7.6 | IC50 | 2 | — | |
ZGDSBEUMPIMXBM
|
7.6 | Ki | 42 | — | |
HPOOZLXEYDPHFI
|
7.6 | IC50 | 3 | — | |
AYJMUFFYIOWRRM
|
7.6 | IC50 | 2 | — | |
BBPZXJMNEQEUBK
|
7.6 | IC50 | 2 | — | |
DTHWSLYDAOOPOE
|
7.6 | IC50 | 4 | — | |
GKMWSAWIKNLTDH
|
7.6 | IC50 | 4 | — | |
MNUPLQVJAOMLAS
|
7.6 | IC50 | 2 | — | |
QDCNDOVOAIZYTL
|
7.6 | IC50 | 4 | — | |
QDCNDOVOAIZYTL
|
7.6 | IC50 | 4 | — | |
CTSDMCNSBRVZGJ
|
7.6 | IC50 | 7 | — | |
DGKPSIOJHHBXOP
|
7.6 | IC50 | 3 | — | |
SLEWGGZPOQNVSU
|
7.6 | IC50 | 22 | — | |
JJXRAZVLEQHSOL
|
7.5 | IC50 | 4 | — | |
RBGSTRWPZHSCTD
|
7.5 | IC50 | 2 | — | |
UFFFDUINWKEBCZ
|
7.5 | IC50 | 2 | — | |
KMDUVZLDXOHFPQ
|
7.5 | IC50 | 4 | — | |
PIRWRQQYRXWTII
|
7.5 | IC50 | 3 | — | |
SFMTZXDPBZEXMO
|
7.5 | IC50 | 2 | — | |
WSTUJEXAPHIEIM
|
7.5 | Kd | 10 | — | |
APLUCVCUSBTPPE
|
7.5 | IC50 | 2 | — | |
DPQDTNJCCOFBNQ
|
7.5 | IC50 | 3 | — | |
FACYQMLOTXHWDQ
|
7.5 | IC50 | 2 | — | |
LLXGNWVOGONTNT
|
7.5 | IC50 | 2 | — | |
GTVWQFJFCAUNFY
|
7.5 | IC50 | 2 | — | |
JREIMVGWCLAHOC
|
7.5 | IC50 | 2 | — | |
LFOWPAZJQIZNHI
|
7.5 | IC50 | 4 | — | |
LFOWPAZJQIZNHI
|
7.5 | IC50 | 4 | — | |
MIYIUVBGBPRNLG
|
7.5 | IC50 | 4 | — | |
NCYONVSVKQVALR
|
7.5 | IC50 | 2 | — | |
YLCUJYLNOPDSFV
|
7.5 | IC50 | 3 | — | |
ZXLFIHLBHMLHFJ
|
7.5 | Ki | 31 | — | |
DGRCFAYRKDYEMX
|
7.5 | IC50 | 7 | — | |
SSISROCLMRBSKK
|
7.5 | IC50 | 2 | — | |
UVBALELUPGCHKQ
|
7.5 | IC50 | 4 | — | |
XWAYWHRXNQJWEN
|
7.5 | IC50 | 3 | — | |
QCLJQTOGBRCCMK
|
7.5 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
7.5 | IC50 | 47 | — | |
OOMBFNDWQIGHEK
|
7.5 | IC50 | 22 | — | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
RROWXJNEWORONQ
|
7.4 | IC50 | 3 | — | |
UHXDASISMPMKEV
|
7.4 | IC50 | 5 | — | |
UZDXOGHTHSYBLJ
|
7.4 | IC50 | 2 | — | |
VPDVHIDCAMWQER
|
7.4 | IC50 | 4 | — | |
OGEBRHQLRGFBNV
|
7.4 | IC50 | 3 | — | |
OGEBRHQLRGFBNV
|
7.4 | IC50 | 3 | — | |
FAILDDCVKDFVJQ
|
7.4 | IC50 | 2 | — | |
GPXJRVLKUZJOES
|
7.4 | IC50 | 3 | — | |
SSWDFFYWXHKOMP
|
7.4 | IC50 | 3 | — | |
VZHCQBXYACZHPJ
|
7.4 | IC50 | 3 | — |