Target Details
| UniProt AC | P30530 |
|---|---|
| Gene Symbol | AXL |
| Protein Name | Tyrosine-protein kinase receptor UFO |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,661
- Clinical molecules 33
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (1,661)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEJGTFPOEJWEGG
|
10.0 | Kd | 149 | — | |
DGVPNVQBSCWKJG
|
10.0 | IC50 | 2 | — | |
ABXVJDAAJIHQCN
|
9.7 | IC50 | 2 | — | |
GFLLLFKVJIGOGF
|
9.7 | IC50 | 2 | — | |
NUQNIAPGIBNTJZ
|
9.7 | IC50 | 2 | — | |
MDPKWYPYSBXZHN
|
9.7 | IC50 | 2 | — | |
FECNHZJRCCTFMT
|
9.5 | IC50 | 2 | — | |
RDKZTOQDJHEFQX
|
9.5 | IC50 | 2 | — | |
PHXDBKCVMGZILA
|
9.4 | IC50 | 2 | — | |
PINVBZQZBYOHQT
|
9.4 | IC50 | 2 | — | |
STZMYLKPKCSIEC
|
9.4 | IC50 | 2 | — | |
VFEZANCUVFZYLF
|
9.4 | IC50 | 2 | — | |
YIFMGCJQLZYTAA
|
9.4 | IC50 | 2 | — | |
VDNNDJSNBJTEFQ
|
9.3 | IC50 | 2 | — | |
WKZAFJWEZVPGCZ
|
9.3 | IC50 | 2 | — | |
XCXMZUYZFOFSTB
|
9.3 | IC50 | 2 | — | |
GEAJYTNNHUHUPD
|
9.2 | IC50 | 2 | — | |
IPHZKBACASVMHL
|
9.2 | IC50 | 2 | — | |
ZSQUNKBTVLUHTH
|
9.2 | IC50 | 2 | — | |
ZYMMXVOIYKLHKH
|
9.2 | IC50 | 2 | — | |
QBRQTJMZEYORSP
|
9.2 | IC50 | 12 | — | |
GFZCTGHGFMTANV
|
9.2 | IC50 | 2 | — | |
HOUOLCBDDCEYMO
|
9.2 | IC50 | 2 | — | |
PBLCTGOWTVQZHF
|
9.2 | IC50 | 2 | — | |
QYCUAHBTLBFVLZ
|
9.2 | IC50 | 2 | — | |
UNWQZQOUOXVJKE
|
9.2 | IC50 | 2 | — | |
WYKOUHBNTYEXKS
|
9.2 | IC50 | 2 | — | |
HJFLVMBTWIJCNF
|
9.1 | IC50 | 3 | — | |
KFASJVNZRIDONN
|
9.1 | IC50 | 2 | — | |
MGUCSMZMGMTIOE
|
9.1 | IC50 | 2 | — | |
OEZCGAGJZUCOEB
|
9.1 | IC50 | 2 | — | |
PKVZAVOIHKTALW
|
9.1 | IC50 | 2 | — | |
SPTBDWLBLZVHRD
|
9.1 | IC50 | 2 | — | |
VKLVODAMMAVNIA
|
9.1 | IC50 | 2 | — | |
WNIAHFXCAWIXLI
|
9.1 | IC50 | 2 | — | |
KGFCIMCRXWIOFT
|
9.1 | IC50 | 2 | — | |
APAJJMXZKHLSSS
|
9.1 | IC50 | 2 | — | |
CZNWNZFIYBTRPU
|
9.1 | IC50 | 2 | — | |
GYWSOFHZIUSHFA
|
9.1 | IC50 | 2 | — | |
ORMXEYBLYMZYLP
|
9.1 | IC50 | 2 | — | |
TXHCXRCHSIVMSN
|
9.1 | IC50 | 3 | — | |
UHQXCBSLWHQJJT
|
9.1 | IC50 | 2 | — | |
JIUGKBKCSODYEF
|
9.0 | IC50 | 2 | — | |
OENGSVYTCJNWNJ
|
9.0 | IC50 | 2 | — | |
SXBRUEVGWHKYKR
|
9.0 | IC50 | 2 | — | |
XGAALYULZCHKHO
|
9.0 | IC50 | 2 | — | |
WVNAHDJJLIHTPX
|
9.0 | IC50 | 2 | — | |
BSDOEKCQNXKTDO
|
9.0 | IC50 | 2 | — | |
LLDHGYBXXLQDJD
|
9.0 | IC50 | 2 | — | |
OAQLTCVWCQRWEW
|
9.0 | IC50 | 2 | — |