Target Details
UniProt ACP29597
Gene SymbolTYK2
Protein NameNon-receptor tyrosine-protein kinase TYK2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1)
Summary
  • Multi-target molecules 3,837
  • Clinical molecules 19
  • Avg pChEMBL 7.56
Top Co-occurrence Targets
Active Molecules (3,837)
InChIKey pChEMBL Type Targets Clinical
LOTLGZUXHGUCOE 9.2 Ki 2
LSAATFWNJDQRQG 9.2 Ki 2
RZTXWBCELPRBKL 9.2 Ki 2
SCWPVGKRRGXLMF 9.2 IC50 4
SMHNRWYUXYBKCG 9.2 Ki 2
VKFCLOVOQMXKJM 9.2 Ki 4
YYUFVSMURUQLMO 9.2 IC50 4
DAYGPXHJOAVVRG 9.2 IC50 4
MSISQTLXMVHCPT 9.2 IC50 4
ULCSWHXDOWVFMK 9.2 IC50 4
VVUPFHUSDJLFEM 9.2 Ki 4
YAHQISLGSOFLRU 9.2 Ki 4
DIBTVUWTGUFWBI 9.2 IC50 4
AOGXHIHTHRCTPK 9.2 Ki 2
CUIBPLIFKMBESI 9.2 Ki 2
FLPXNQWEAODYRF 9.2 Ki 2
HABNRCDBMMDTDR 9.2 Ki 2
HROWLWGDTOBEDM 9.2 Ki 2
JBYYBYKZQWGOJL 9.2 Ki 2
RATPMJAJYLJWHS 9.2 Ki 2
SHSAMLWCDMVMLO 9.2 Ki 3
UZUOFBYCMXECPS 9.2 Ki 2
VRYUZSRAENQEKH 9.2 IC50 4
YXKUPJSJNAKRLQ 9.2 Ki 2
ZFFSYYHNBNAIRW 9.2 Ki 2
BPDXDZDEFQATRW 9.2 IC50 4
WZCAXUNOMZZMQX 9.2 IC50 2
AVRFACACEWCPRC 9.2 IC50 4
AQSSMEORRLJZLU 9.2 Kd 34 Yes
DFZGJZRKSHDCMG 9.2 IC50 4
HQUBADRFDQYRJZ 9.2 IC50 4
JKESNMWWWWZHEN 9.2 IC50 4
KLPJBSUBJNVPFZ 9.2 IC50 4
MFANTCFRQWVMFZ 9.2 IC50 2
MWEQLWHNRFPCEW 9.2 Ki 2
OANXOEXNBCTCLW 9.2 Ki 2
YFSPSGACYXXNNF 9.2 Ki 6
YFZKQJYONASWFW 9.2 IC50 7
DCAHNNRXGSGGCL 9.1 IC50 4
VZMBJDMHDUJNSV 9.1 IC50 4
JMGHYHLHFYFKKM 9.1 IC50 4
DIUNXEXOCMDGQL 9.1 IC50 3
JIQQEQXPBPQIPX 9.1 IC50 4
KAVVKRQBEAWLIE 9.1 Ki 4
KZPCATSDOZHYDA 9.1 Ki 4
RINWDSCUVKTALQ 9.1 Ki 4
SCFXRVXGXNBVDI 9.1 IC50 3
SYMXGYXFLGDULR 9.1 IC50 4
UIICOJMWXQEEML 9.1 Ki 2
VMLVHRAAZGJBIV 9.1 IC50 4
2D structure