Target Details
| UniProt AC | P29597 |
|---|---|
| Gene Symbol | TYK2 |
| Protein Name | Non-receptor tyrosine-protein kinase TYK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 3,837
- Clinical molecules 19
- Avg pChEMBL 7.56
KEGG Pathways (17)
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- NOD-like receptor signaling pathway
- Necroptosis
- Osteoclast differentiation
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Toll-like receptor signaling pathway
- Toxoplasmosis
Associated Diseases (2)
Active Molecules (3,837)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JNOPCQSOHNYICW
|
9.8 | IC50 | 4 | — | |
SPQRBCVHNZXRER
|
9.8 | IC50 | 2 | — | |
TYZYHIAKKRJCBW
|
9.7 | Kd | 2 | — | |
BNOPEBHGDTWAQX
|
9.7 | IC50 | 4 | — | |
ALTZMYUVVKYDIX
|
9.7 | IC50 | 2 | — | |
BFBCSHXBVZNRRU
|
9.7 | IC50 | 2 | — | |
IKSRDHMMQOCRHN
|
9.7 | IC50 | 4 | — | |
IKURBZUUPLCTRI
|
9.7 | IC50 | 4 | — | |
KZBPYAFBSQFJHT
|
9.7 | IC50 | 2 | — | |
LTRURJCNQJXBNG
|
9.7 | IC50 | 4 | — | |
NWPDHXISBFEDSN
|
9.7 | IC50 | 2 | — | |
OGYDMBQWFWOTHF
|
9.7 | IC50 | 3 | — | |
PVSLHTFARDGGLL
|
9.7 | IC50 | 4 | — | |
UDGMZRVCKLNKHN
|
9.7 | IC50 | 3 | — | |
XIZMNLZDSOAQFL
|
9.7 | IC50 | 2 | — | |
YAHGUPVIQAEPKI
|
9.7 | IC50 | 4 | — | |
BCMIRTHEUWYNHX
|
9.7 | IC50 | 4 | — | |
KEIGGTSBOIAQRO
|
9.7 | IC50 | 2 | — | |
WRFANJMETRKSFA
|
9.7 | IC50 | 4 | — | |
LJGKJOABCDCQLE
|
9.6 | IC50 | 4 | — | |
LNTSTFPYHHHPLZ
|
9.6 | IC50 | 4 | — | |
PMCNHBRGNUQKHF
|
9.6 | IC50 | 4 | — | |
FIXODQLYPRSTCO
|
9.6 | Ki | 4 | — | |
FIXODQLYPRSTCO
|
9.6 | Ki | 4 | — | |
PLOAUINIELSVFC
|
9.6 | Ki | 4 | — | |
UAHMLABNZNESHG
|
9.6 | IC50 | 7 | — | |
NRYOXXMMQVNECT
|
9.6 | IC50 | 4 | — | |
FPLDLCFSEQHYEF
|
9.6 | IC50 | 4 | — | |
BKLNXXJBSLIJFP
|
9.5 | IC50 | 2 | — | |
QIUJVZGYISFYIX
|
9.5 | IC50 | 3 | — | |
BWEHAWAXNXZSRX
|
9.5 | IC50 | 2 | — | |
DPDKHLQHVXKOQW
|
9.5 | IC50 | 2 | — | |
GLASCLXQTDIOAT
|
9.5 | IC50 | 2 | — | |
GYBXQCLWSUJTMN
|
9.5 | Ki | 2 | — | |
IRIDDEHSOPFQKO
|
9.5 | IC50 | 4 | — | |
OULORHJOSYJPAD
|
9.5 | IC50 | 4 | — | |
ROTAUGLEOWMJMR
|
9.5 | IC50 | 3 | — | |
CHUJALYWQZENTG
|
9.5 | IC50 | 4 | — | |
KAHARENCCCTWSQ
|
9.5 | Ki | 4 | — | |
LKYNKWVSJBBRNP
|
9.5 | Ki | 4 | — | |
VERYIUBILUMSSE
|
9.5 | IC50 | 4 | — | |
VLAHIKLMFQZDPR
|
9.5 | IC50 | 4 | — | |
GVZIGWRNCRFSBD
|
9.5 | IC50 | 2 | — | |
UWCJNDNJYBLIQE
|
9.5 | IC50 | 4 | — | |
VTOHXCTUKVQTFB
|
9.4 | IC50 | 4 | — | |
XQZMCWSNDJGPHN
|
9.4 | IC50 | 4 | — | |
IRIDDEHSOPFQKO
|
9.4 | IC50 | 4 | — | |
LSQWGVOEBUCSKN
|
9.4 | IC50 | 4 | — | |
QNWIWKOFJUZOHT
|
9.4 | IC50 | 2 | — | |
IPWDOXJGNQLPOD
|
9.4 | IC50 | 2 | — |