Target Details
| UniProt AC | P29597 |
|---|---|
| Gene Symbol | TYK2 |
| Protein Name | Non-receptor tyrosine-protein kinase TYK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 3,837
- Clinical molecules 19
- Avg pChEMBL 7.56
KEGG Pathways (17)
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- NOD-like receptor signaling pathway
- Necroptosis
- Osteoclast differentiation
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Toll-like receptor signaling pathway
- Toxoplasmosis
Associated Diseases (2)
Active Molecules (3,837)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XRWOEOJYJUHVML
|
8.5 | IC50 | 4 | — | |
FMJVBOXWJGDNJK
|
8.5 | IC50 | 4 | — | |
NAXUVOPYFVMTNB
|
8.5 | IC50 | 4 | — | |
PCIVQDNLJCQJCG
|
8.5 | IC50 | 4 | — | |
LTGGHOLQJAWCLY
|
8.4 | IC50 | 4 | — | |
DRRPDXUMHCIICI
|
8.4 | IC50 | 4 | — | |
UEFBECCKJTVZES
|
8.4 | IC50 | 4 | — | |
UXEHANJJLFQUIY
|
8.4 | IC50 | 4 | — | |
VDAREBZGZZDSKX
|
8.4 | IC50 | 4 | — | |
CUOWQRBLXGZKTO
|
8.4 | IC50 | 4 | — | |
CWGBVVJEMFFMQL
|
8.4 | IC50 | 2 | — | |
JRUFFDAPSGAZIL
|
8.4 | IC50 | 4 | — | |
QXRSSWDWVCPRRK
|
8.4 | IC50 | 2 | — | |
VBWXTYCDRUUVPK
|
8.4 | IC50 | 4 | — | |
BJIMEBGDCGRSIB
|
8.4 | IC50 | 4 | — | |
DDMBPFJHFQVXGI
|
8.4 | IC50 | 2 | — | |
JFEOTMHLMSEPBP
|
8.4 | IC50 | 4 | — | |
VCJNQQKABAEVLV
|
8.4 | IC50 | 4 | — | |
YRAPEEGRAZXEHV
|
8.4 | IC50 | 4 | — | |
ZFGRPZIMBQPZJH
|
8.4 | IC50 | 4 | — | |
CCMBJIATBMXYFC
|
8.4 | IC50 | 4 | — | |
CQZQKLHERRXFEZ
|
8.4 | IC50 | 4 | — | |
SJXBCXWWUGDWBF
|
8.4 | IC50 | 4 | — | |
YKTYTOSJOTWOCE
|
8.4 | IC50 | 4 | — | |
ZSTUJCOZGCERSU
|
8.4 | IC50 | 4 | — | |
CEXXEJLTBYXKAX
|
8.4 | IC50 | 3 | — | |
JVJZKTVGPRSEMX
|
8.4 | IC50 | 4 | — | |
LRJHFOMJPOSHDU
|
8.4 | IC50 | 4 | — | |
LWHQMSMLWVYUDX
|
8.4 | IC50 | 2 | — | |
QZUWXMXRQHXTOB
|
8.4 | IC50 | 3 | — | |
WHQSFRQPKNDBED
|
8.4 | IC50 | 2 | — | |
XHIOCQXKIGYBIL
|
8.4 | IC50 | 4 | — | |
ZFEDARIKGLHKFD
|
8.4 | IC50 | 4 | — | |
ZXAFLEVWBXJCQF
|
8.4 | IC50 | 6 | — | |
BGKOWTMJBZMFDL
|
8.4 | IC50 | 2 | — | |
MHXZXPSUUPWZDU
|
8.4 | IC50 | 4 | — | |
MHXZXPSUUPWZDU
|
8.4 | IC50 | 4 | — | |
QOSFYCUGTCNTRN
|
8.4 | IC50 | 4 | — | |
RORMJCXVRLHBIE
|
8.4 | IC50 | 4 | — | |
URVFJVXEAYRVCV
|
8.4 | Ki | 4 | — | |
CSKWMCUZWIEQHE
|
8.4 | IC50 | 2 | — | |
LMWQAELGOVWZFY
|
8.4 | IC50 | 4 | — | |
NVFYPSBGYRSLQB
|
8.4 | IC50 | 4 | — | |
SZWULWDUCCLMJA
|
8.4 | Ki | 4 | — | |
VEPPHPJVFXUYOF
|
8.4 | IC50 | 4 | — | |
XUZJGEGSRPWEIU
|
8.4 | IC50 | 4 | — | |
MPUPFFCJTANSDV
|
8.4 | IC50 | 4 | — | |
MXZNRXIGJIAJNT
|
8.4 | IC50 | 4 | — | |
NLGZSRKKPYFWHZ
|
8.4 | IC50 | 6 | — | |
NLVCYHWVVMCSAF
|
8.4 | IC50 | 4 | — |