Target Details
| UniProt AC | P29597 |
|---|---|
| Gene Symbol | TYK2 |
| Protein Name | Non-receptor tyrosine-protein kinase TYK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 3,837
- Clinical molecules 19
- Avg pChEMBL 7.56
KEGG Pathways (17)
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- NOD-like receptor signaling pathway
- Necroptosis
- Osteoclast differentiation
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Toll-like receptor signaling pathway
- Toxoplasmosis
Associated Diseases (2)
Active Molecules (3,837)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XOBYWVCCKFXUKO
|
8.6 | IC50 | 4 | — | |
BYJBWSMAHQTPCB
|
8.6 | IC50 | 4 | — | |
DZUSPKFBRQRYNR
|
8.6 | IC50 | 5 | — | |
FBMPIPDDIOMXIM
|
8.6 | IC50 | 4 | — | |
FVWPSGHGQQMRKR
|
8.6 | IC50 | 4 | — | |
LUAWBDVVBXMLEL
|
8.6 | IC50 | 7 | — | |
MTLAJFMANDWYIE
|
8.6 | IC50 | 4 | — | |
OTAWEODWHFBSCD
|
8.6 | IC50 | 4 | — | |
PPDRYWDVANCHFT
|
8.6 | IC50 | 4 | — | |
PXALDOWLQORFBK
|
8.6 | IC50 | 4 | — | |
WVYXBGBSMGFRJF
|
8.6 | IC50 | 4 | — | |
CENFCEFROIFFFD
|
8.5 | IC50 | 4 | — | |
FJVHUAHOQGQJNZ
|
8.5 | IC50 | 4 | — | |
FZXMPCXMYBNDEB
|
8.5 | IC50 | 4 | — | |
MDTIFFXIWIDZBH
|
8.5 | IC50 | 4 | — | |
OQNGITUNHHCSOA
|
8.5 | IC50 | 4 | — | |
SRVNAKKCHOGLQU
|
8.5 | IC50 | 3 | — | |
VGBYAYCYPVFDTM
|
8.5 | IC50 | 6 | — | |
FNVZUMZCEAGHIK
|
8.5 | IC50 | 4 | — | |
GGUONJQHHUWSQC
|
8.5 | IC50 | 4 | — | |
KJSACPRRGVARJC
|
8.5 | IC50 | 6 | — | |
LSJQWYSSWDBQHW
|
8.5 | IC50 | 4 | — | |
LSPIMHPSWRNVOM
|
8.5 | IC50 | 3 | — | |
MKQFWNKDBIRKBB
|
8.5 | IC50 | 3 | — | |
RZVBCGFEXPDAAN
|
8.5 | IC50 | 4 | — | |
YESOLTRAONBOKK
|
8.5 | Kd | 2 | — | |
GNVJDFYURAVLOR
|
8.5 | IC50 | 3 | — | |
VWVYILCFSYNJHF
|
8.5 | Ki | 49 | — | |
WPKFVOMIANZVBJ
|
8.5 | IC50 | 4 | — | |
RLMMSHIOBVKROE
|
8.5 | IC50 | 4 | — | |
UKXSXAADXKCVTQ
|
8.5 | IC50 | 4 | — | |
ZCDNUYKDPDTEOY
|
8.5 | IC50 | 2 | — | |
ZMWNZVPHESZOJV
|
8.5 | Ki | 2 | — | |
DGDMQGMQJGOQNY
|
8.5 | IC50 | 2 | — | |
DYCFJMLAPBEYRV
|
8.5 | IC50 | 4 | — | |
MLITXGDEKAPRNU
|
8.5 | IC50 | 4 | — | |
QATVMVPAHQPMOK
|
8.5 | IC50 | 4 | — | |
ROCWQSCNNATQOY
|
8.5 | IC50 | 4 | — | |
UOSGIRBXSBYVHS
|
8.5 | IC50 | 4 | — | |
USVKVOHLTFMVFN
|
8.5 | IC50 | 4 | — | |
VGQGFYCOZCNACG
|
8.5 | IC50 | 4 | — | |
ZLZPLFCWNAIVRT
|
8.5 | IC50 | 4 | — | |
ZRWAPJQBKMIZOF
|
8.5 | IC50 | 4 | — | |
HIXYDBSLZYKHEU
|
8.5 | Ki | 3 | — | |
JNUDIJJVTYHAPN
|
8.5 | IC50 | 4 | — | |
OTPVYQFYPRLIGT
|
8.5 | Kd | 2 | — | |
QLPWFQPHRAFDGC
|
8.5 | IC50 | 7 | — | |
SBXSPNBGVSORJP
|
8.5 | IC50 | 4 | — | |
UXRAMPPWHJVSRI
|
8.5 | IC50 | 4 | — | |
VYUZMRQDNWEZOD
|
8.5 | IC50 | 5 | — |