Target Details
| UniProt AC | P29597 |
|---|---|
| Gene Symbol | TYK2 |
| Protein Name | Non-receptor tyrosine-protein kinase TYK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1) |
Summary
- Multi-target molecules 3,837
- Clinical molecules 19
- Avg pChEMBL 7.56
KEGG Pathways (17)
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- NOD-like receptor signaling pathway
- Necroptosis
- Osteoclast differentiation
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Toll-like receptor signaling pathway
- Toxoplasmosis
Associated Diseases (2)
Active Molecules (3,837)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQDKZKSLBHKUGR
|
8.8 | IC50 | 4 | — | |
KQAJQVQIWBQIFM
|
8.8 | IC50 | 4 | — | |
NKALKXMQBFLGQI
|
8.8 | Ki | 2 | — | |
OOMAPNJTWLGJDI
|
8.8 | Ki | 2 | — | |
WPFTYCRFFPGAGZ
|
8.8 | IC50 | 4 | — | |
RIWJSTAVOOCXPT
|
8.8 | IC50 | 3 | — | |
DDDCWZSEFHBEGC
|
8.8 | IC50 | 4 | — | |
BYXNEKGOGSKHAW
|
8.8 | IC50 | 4 | — | |
LLRNGFSFYHDPKW
|
8.8 | Ki | 3 | — | |
OFPQQEBBZKPLFE
|
8.8 | Ki | 2 | — | |
XQDJIZPXYHDJDG
|
8.8 | IC50 | 3 | — | |
BRIUDIRHWGESSC
|
8.8 | IC50 | 4 | — | |
GLXJKUDCHGMWME
|
8.8 | IC50 | 4 | — | |
PMOCYAUOLYFXTN
|
8.8 | IC50 | 4 | — | |
BOWWMYAPYXYIJF
|
8.7 | Ki | 2 | — | |
CYFYEGKSPAEQGC
|
8.7 | IC50 | 4 | — | |
DABPGIDEMDQWKD
|
8.7 | IC50 | 2 | — | |
GEQOWUCLQGOQHZ
|
8.7 | IC50 | 4 | — | |
HBOBPFABMCQOIY
|
8.7 | IC50 | 4 | — | |
HSPSGYMCTYNNSC
|
8.7 | IC50 | 4 | — | |
JYCAAJPPOBUPNX
|
8.7 | IC50 | 4 | — | |
WZJIVMCLVPKPHR
|
8.7 | IC50 | 4 | — | |
OZDFKECLFIDGPK
|
8.7 | IC50 | 4 | — | |
VTHLBHXTIANZQX
|
8.7 | IC50 | 4 | — | |
FETNQDDVHOUWMB
|
8.7 | IC50 | 4 | — | |
ITHVYCKTQCDGNM
|
8.7 | IC50 | 3 | — | |
MOZBSVJPDSKZMY
|
8.7 | IC50 | 4 | — | |
QBMBKEGWVSJZNL
|
8.7 | IC50 | 4 | — | |
QFUPNRFOUYLYGG
|
8.7 | IC50 | 4 | — | |
ZPBRNDUJNKMEMH
|
8.7 | Kd | 3 | — | |
IUVVBOQAVMSUQH
|
8.7 | IC50 | 3 | — | |
WNRXTALSWGUQLZ
|
8.7 | IC50 | 4 | — | |
BNXOIVMMIFOVPX
|
8.7 | IC50 | 3 | — | |
BZZKEPGENYLQSC
|
8.7 | IC50 | 6 | — | |
DHWQGOLXINKFNQ
|
8.7 | IC50 | 4 | — | |
GKHBPPWDKONWDH
|
8.7 | IC50 | 4 | — | |
IBJWEQLGJBSZHA
|
8.7 | IC50 | 2 | — | |
JONZPWSVTNTRMO
|
8.7 | IC50 | 2 | — | |
JXLWZLUHIKGJID
|
8.7 | IC50 | 4 | — | |
JXLWZLUHIKGJID
|
8.7 | IC50 | 4 | — | |
KCNDGFPTNZEEGQ
|
8.7 | IC50 | 2 | — | |
LWMFNMXXGFQOGG
|
8.7 | IC50 | 4 | — | |
OYFHYNGYRZEOJP
|
8.7 | IC50 | 3 | — | |
PDOQBOJDRPLBQU
|
8.7 | IC50 | 21 | — | |
PMXSQTYWBDXQET
|
8.7 | IC50 | 4 | — | |
QLSJFVSWCVEOMO
|
8.7 | IC50 | 4 | — | |
RJHREQOUJMQXBL
|
8.7 | IC50 | 4 | — | |
UPBRYBJZTWHUQK
|
8.7 | IC50 | 4 | — | |
VAMHUIZQIUMVCB
|
8.7 | IC50 | 4 | — | |
VWCMCKGLNBSIAJ
|
8.7 | IC50 | 2 | — |