Target Details
| UniProt AC | P29466 |
|---|---|
| Gene Symbol | CASP1 |
| Protein Name | Caspase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00619 (CARD) PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 173
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (16)
- Amyotrophic lateral sclerosis
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Influenza A
- Legionellosis
- Lipid and atherosclerosis
- NOD-like receptor signaling pathway
- Necroptosis
- Neutrophil extracellular trap formation
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Shigellosis
- Yersinia infection
Active Molecules (173)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADCRWKOZMQLEEC
|
6.3 | Ki | 3 | — | |
ZUMYWWOOYMHLPE
|
6.3 | IC50 | 2 | — | |
DOIAAMNEXGWYFQ
|
6.2 | IC50 | 2 | — | |
UVJNVVPTQWFZMT
|
6.2 | IC50 | 4 | — | |
KYPWBBBOBAOGSQ
|
6.2 | IC50 | 2 | — | |
NERMQYMDDXNPRD
|
6.2 | IC50 | 2 | — | |
ZPGKPGJAPADYFS
|
6.2 | Ki | 2 | — | |
RVUPUUXSFOLOAS
|
6.2 | IC50 | 3 | — | |
ABCKZNSVBLCRMS
|
6.2 | IC50 | 3 | — | |
LPQLYZKOKVZVSN
|
6.2 | IC50 | 4 | — | |
LPQLYZKOKVZVSN
|
6.2 | IC50 | 4 | — | |
VFANYHPZKZVWGL
|
6.2 | IC50 | 2 | — | |
WIYBIQZLIVGWQF
|
6.2 | IC50 | 3 | — | |
WUQPWSWGFKLLRA
|
6.2 | IC50 | 2 | — | |
BVAULMYVOSWSBQ
|
6.1 | IC50 | 2 | — | |
JMCSMHDKXZIFQR
|
6.1 | IC50 | 4 | — | |
XXQCRRRNRLLOKC
|
6.1 | IC50 | 2 | — | |
IBUIGAOZEYCWCZ
|
6.1 | IC50 | 2 | — | |
PKCZPKXBVIXOLU
|
6.1 | IC50 | 2 | — | |
YDWMZYBWKLFQKO
|
6.1 | IC50 | 3 | — | |
DPHACENAZHGWHS
|
6.0 | IC50 | 4 | — | |
DTFCKUHAUSPAPY
|
6.0 | Ki | 2 | — | |
UPNDCXMMARFRPM
|
6.0 | IC50 | 3 | — |