Target Details
| UniProt AC | P29466 |
|---|---|
| Gene Symbol | CASP1 |
| Protein Name | Caspase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00619 (CARD) PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 173
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (16)
- Amyotrophic lateral sclerosis
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Influenza A
- Legionellosis
- Lipid and atherosclerosis
- NOD-like receptor signaling pathway
- Necroptosis
- Neutrophil extracellular trap formation
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Shigellosis
- Yersinia infection
Active Molecules (173)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RIHVWVMASFXAPK
|
7.5 | IC50 | 2 | — | |
GFJVEQNTNYTSIH
|
7.4 | IC50 | 2 | — | |
KQJSQWZMSAGSHN
|
7.4 | IC50 | 9 | — | |
RYTHJGWSBNDVTE
|
7.4 | IC50 | 2 | — | |
HZSYROXMXVMKLR
|
7.4 | Ki | 2 | — | |
NHIDZXMAMOZUNW
|
7.4 | IC50 | 3 | — | |
UCWNTWGHVCSMJP
|
7.3 | IC50 | 2 | — | |
BFIRSNDOLOQSCL
|
7.3 | IC50 | 2 | — | |
CYHOOSOSVKYWRO
|
7.3 | IC50 | 2 | — | |
IJQPLPVGYLMXIU
|
7.3 | IC50 | 2 | — | |
INEQQSYFBJJTKI
|
7.3 | IC50 | 5 | — | |
LBGLGTAQLROFTM
|
7.3 | Ki | 3 | — | |
SCUZVSHLJVHGDP
|
7.3 | Ki | 3 | — | |
SKSZJGAFHISZNB
|
7.3 | IC50 | 5 | — | |
XIMITGPWYYFUQF
|
7.3 | IC50 | 5 | — | |
ZMIXZDFAIQPNIS
|
7.3 | IC50 | 3 | — | |
JFACETXYABVHFD
|
7.2 | IC50 | 2 | — | |
CIDFSOFEWVUWHQ
|
7.2 | IC50 | 4 | — | |
XIMITGPWYYFUQF
|
7.2 | IC50 | 3 | — | |
HHHCHMWEUVMQER
|
7.1 | IC50 | 4 | — | |
HHHCHMWEUVMQER
|
7.1 | IC50 | 4 | — | |
LZSIDSOVZDJMCX
|
7.0 | IC50 | 3 | — | |
PABZSOUNSSUXIN
|
7.0 | Ki | 2 | — | |
YNRQFMSSDVQNGQ
|
7.0 | IC50 | 5 | — | |
ZJZZXNFEARKFRC
|
7.0 | IC50 | 3 | — | |
WLZOCGMSLPOOIC
|
6.9 | IC50 | 4 | — | |
NCLFPGSWIDLTSV
|
6.8 | IC50 | 2 | — | |
ZHVMILHEPYUCKZ
|
6.8 | IC50 | 3 | — | |
FMTZTJFXNZOBIQ
|
6.8 | Ki | 5 | — | |
UMBVAPCONCILTL
|
6.7 | IC50 | 5 | — | |
KQLWSSDYPGXCNL
|
6.6 | IC50 | 3 | — | |
XTPTVAPEXHUUDR
|
6.6 | IC50 | 3 | — | |
RVAGESXTEHAWEY
|
6.5 | Ki | 3 | — | |
ZSOPKWJQJKUHFH
|
6.5 | IC50 | 2 | — | |
DWGRSJBIHVFBFL
|
6.5 | IC50 | 3 | — | |
KACACYYTPVUKSL
|
6.5 | IC50 | 2 | — | |
LDDAWLZYJRJPPR
|
6.5 | IC50 | 4 | — | |
VIUJQQJJJZNKDP
|
6.5 | IC50 | 4 | — | |
LTBPAHIEHDBOIC
|
6.5 | IC50 | 2 | — | |
UTNIELHSQXTLFN
|
6.5 | IC50 | 3 | — | |
HSCFCMDPCFLHTC
|
6.4 | IC50 | 2 | — | |
AOUFLZQXBYFGOZ
|
6.4 | IC50 | 3 | — | |
TWGFWBPIHYEITI
|
6.4 | IC50 | 2 | — | |
MFHQDLHNUMVDLA
|
6.4 | IC50 | 4 | — | |
KGHGMUBHFANXGE
|
6.4 | IC50 | 2 | — | |
QLHHECDAKBHQND
|
6.4 | IC50 | 2 | — | |
ZEWZRCNXHOUXDN
|
6.4 | IC50 | 3 | — | |
CEFXQYILQBZDCM
|
6.3 | IC50 | 2 | — | |
VZUJUIONFIJSIE
|
6.3 | IC50 | 3 | — | |
YMYGKHWZVMKILN
|
6.3 | IC50 | 2 | — |