Target Details
| UniProt AC | P29466 |
|---|---|
| Gene Symbol | CASP1 |
| Protein Name | Caspase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00619 (CARD) PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 173
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (16)
- Amyotrophic lateral sclerosis
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Influenza A
- Legionellosis
- Lipid and atherosclerosis
- NOD-like receptor signaling pathway
- Necroptosis
- Neutrophil extracellular trap formation
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Shigellosis
- Yersinia infection
Active Molecules (173)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UUEMWRIOZLIPHU
|
8.5 | IC50 | 4 | — | |
CKRCPAGGKUFVIT
|
8.5 | IC50 | 4 | — | |
MTGSTDMYYFQKEE
|
8.5 | IC50 | 3 | — | |
CXAGHAZMQSCAKJ
|
8.4 | IC50 | 2 | — | |
JEYQBANFJYIELI
|
8.4 | IC50 | 4 | — | |
LVXZMAMJNHAXKU
|
8.4 | IC50 | 4 | — | |
BPPAKSZSGBPOEH
|
8.3 | IC50 | 4 | — | |
IMKLAZABQHZAJN
|
8.3 | IC50 | 2 | — | |
IOVDCXCEGWOHSX
|
8.3 | IC50 | 2 | — | |
YSDNTHYUFYFOEN
|
8.3 | IC50 | 4 | — | |
HBVXRUIPTGRFDT
|
8.2 | IC50 | 2 | — | |
MBPKVWLXSMFUMN
|
8.2 | IC50 | 4 | — | |
YBUQKGADXMDZCC
|
8.2 | IC50 | 2 | — | |
DOBIYIOPZIMMRH
|
8.2 | Ki | 3 | — | |
NETBIBQTHPVZHP
|
8.2 | IC50 | 4 | — | |
SCZQZYJOIBQIGS
|
8.2 | IC50 | 4 | — | |
ULELQXPHOSNTHT
|
8.2 | IC50 | 4 | — | |
XMHRXPMKDALTSG
|
8.2 | IC50 | 2 | — | |
GEZSSSVQIGDDMR
|
8.1 | IC50 | 4 | — | |
PCKDUAQUKNXESJ
|
8.1 | IC50 | 4 | — | |
PSEYKDQFSOGYNR
|
8.1 | IC50 | 4 | — | |
ZXYUJUZVJDHMDR
|
8.0 | IC50 | 4 | — | |
NHHJXCJHJPGPEF
|
8.0 | IC50 | 4 | — | |
DGOJTUAQSDYETG
|
8.0 | IC50 | 2 | — | |
SIQQBFWEHZXLAO
|
7.9 | IC50 | 6 | — | |
QLHDEYZCVHOGEF
|
7.9 | IC50 | 4 | — | |
CBORVVSGKICHTH
|
7.9 | IC50 | 2 | — | |
AFVSWIIKNZNPMC
|
7.8 | IC50 | 2 | — | |
NCCIOJYCWRHZMY
|
7.8 | IC50 | 4 | — | |
LRHHFDQCXBPQLY
|
7.8 | IC50 | 7 | — | |
YAXZZOWMNVKCTF
|
7.8 | IC50 | 2 | — | |
ZYWFKPCNVPPHDB
|
7.8 | IC50 | 2 | — | |
BAHXAEZPSDVZAI
|
7.7 | Ki | 2 | — | |
QHMBSVQNZZTUGM
|
7.7 | Kd | 13 | — | |
NJAQASWTRGUAGC
|
7.7 | IC50 | 3 | — | |
SVQAMGNGTJSUFV
|
7.7 | IC50 | 3 | — | |
FJKDUHWEJJLMQP
|
7.7 | IC50 | 3 | — | |
LYBWGROBJJXCJJ
|
7.7 | IC50 | 6 | — | |
NAZSWKZWCFVHEL
|
7.7 | IC50 | 4 | — | |
IMRNKNWXBGSFOO
|
7.7 | IC50 | 2 | — | |
ZFUKMGBZRXETJQ
|
7.6 | IC50 | 3 | — | |
NFNHDUDACIDJAE
|
7.6 | IC50 | 3 | — | |
NFNHDUDACIDJAE
|
7.6 | IC50 | 3 | — | |
UUTWTWROPLXGDT
|
7.5 | IC50 | 3 | — | |
XIMSCIZHMWOJHC
|
7.5 | IC50 | 3 | — | |
HIBILFREOVFCHQ
|
7.5 | IC50 | 4 | — | |
GRTICURLEQIPRO
|
7.5 | IC50 | 3 | — | |
JPCVJWQLKRHLRX
|
7.5 | IC50 | 3 | — | |
WPBCCSIRQOJBIN
|
7.5 | IC50 | 3 | — | |
NUEXSSWTCJYNJY
|
7.5 | IC50 | 4 | — |