Target Details
| UniProt AC | P29466 |
|---|---|
| Gene Symbol | CASP1 |
| Protein Name | Caspase-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00619 (CARD) PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 173
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (16)
- Amyotrophic lateral sclerosis
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Influenza A
- Legionellosis
- Lipid and atherosclerosis
- NOD-like receptor signaling pathway
- Necroptosis
- Neutrophil extracellular trap formation
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Shigellosis
- Yersinia infection
Active Molecules (173)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XIMITGPWYYFUQF
|
10.3 | IC50 | 8 | — | |
YNRQFMSSDVQNGQ
|
10.0 | IC50 | 8 | — | |
HDXDXAKYCMKPSF
|
9.6 | IC50 | 4 | — | |
MDRQEFUKIMUQFX
|
9.4 | IC50 | 4 | — | |
QFAGZHXWKDBXGQ
|
9.1 | IC50 | 4 | — | |
UCOGGEXRPKAPHO
|
9.1 | IC50 | 3 | — | |
GQDJBEWJIKPEQS
|
9.1 | IC50 | 3 | — | |
CSEDBYKWGJUWMQ
|
9.0 | IC50 | 3 | — | |
ASXOTWMUUUHDST
|
9.0 | IC50 | 2 | — | |
CBORVVSGKICHTH
|
9.0 | IC50 | 2 | — | |
ITXGNTGSRFVVNR
|
9.0 | IC50 | 2 | — | |
JSLLIKPZGONZEJ
|
9.0 | IC50 | 2 | — | |
KXAUXHBXAIZBIR
|
9.0 | Ki | 2 | — | |
METJQQYBQDJDER
|
9.0 | IC50 | 2 | — | |
OEMJCZSXKAMRQI
|
9.0 | IC50 | 2 | — | |
OHCGXQWQIAAFLW
|
9.0 | IC50 | 2 | — | |
QPXWSOVNNLBWQP
|
9.0 | IC50 | 2 | — | |
RHMWMZJZYRGSKL
|
9.0 | IC50 | 2 | — | |
VURUGTWAAZWTEC
|
9.0 | IC50 | 2 | — | |
WNMPCOLHJBPQIT
|
9.0 | IC50 | 2 | — | |
XQDAIAVDJUUPEN
|
9.0 | IC50 | 2 | — | |
XQRCYZUOALTFCB
|
9.0 | IC50 | 2 | — | |
YIKMAFZEIMZOGL
|
9.0 | Ki | 2 | — | |
YPSFOQSJNMXHOO
|
9.0 | IC50 | 2 | — | |
ZJOMIVVGRLRQHB
|
9.0 | IC50 | 2 | — | |
MPIKODMIUDLWKY
|
9.0 | IC50 | 3 | — | |
SDUIHZXGXLYNPJ
|
9.0 | IC50 | 2 | — | |
VBXOCZFAWPHIJQ
|
9.0 | IC50 | 3 | — | |
SHHIOGGLCRQOHT
|
8.9 | IC50 | 4 | — | |
ORBZCGMLHAHSPL
|
8.9 | IC50 | 2 | — | |
UWYWIWOJPZFFAT
|
8.8 | IC50 | 4 | — | |
GGRODTCKLDDOBP
|
8.8 | IC50 | 3 | — | |
JYGKCHPWCXRSQJ
|
8.8 | IC50 | 4 | — | |
KSIBLECLZAACGQ
|
8.8 | IC50 | 3 | — | |
MNAXVQLJZGETJF
|
8.8 | IC50 | 3 | — | |
IYUHLZOWOKCWMK
|
8.7 | IC50 | 3 | — | |
VIKAKOARTUQKPC
|
8.7 | IC50 | 3 | — | |
GCDOZFZRBUNMDE
|
8.7 | IC50 | 3 | — | |
WZRDTXYFPUFFST
|
8.7 | IC50 | 3 | — | |
XWTJWAAMOCNKHH
|
8.7 | IC50 | 4 | — | |
GPEBKBVTPDFRPO
|
8.7 | IC50 | 2 | — | |
QAFBFHNIUINEJN
|
8.7 | IC50 | 4 | — | |
SHDGJJPFMISTHO
|
8.7 | IC50 | 4 | — | |
YEUTYABUIBVFMW
|
8.7 | IC50 | 2 | — | |
DONUNLOVYIQJNS
|
8.7 | IC50 | 4 | — | |
INTJRTIYLCEHRJ
|
8.7 | IC50 | 4 | — | |
SFDIMTVHWVLTIP
|
8.7 | IC50 | 4 | — | |
BTAFTKGHXXQLHC
|
8.6 | IC50 | 4 | — | |
UIYYZKYDLKUXII
|
8.5 | IC50 | 2 | — | |
UUEMWRIOZLIPHU
|
8.5 | IC50 | 4 | — |