Target Details
| UniProt AC | P29376 |
|---|---|
| Gene Symbol | LTK |
| Protein Name | Leukocyte tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 127
- Clinical molecules 16
- Avg pChEMBL 7.0
Active Molecules (127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UHTHHESEBZOYNR
|
6.3 | Kd | 66 | Yes | |
BIIVYFLTOXDAOV
|
6.2 | Ki | 31 | — | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
IJRBJCMLWLFMIN
|
6.2 | Ki | 17 | — | |
KDJGCVHPUMHUOL
|
6.2 | Ki | 11 | — | |
NOBMKUVHFRVBES
|
6.2 | Ki | 19 | — | |
UGUZOLHBLLTLBA
|
6.2 | Ki | 15 | — | |
YYPKOMNJRZRWIC
|
6.2 | Ki | 26 | — | |
CJUJLGFTKBBDMG
|
6.1 | Ki | 9 | — | |
DVWFMBFZDOBWAD
|
6.1 | Ki | 8 | — | |
GZAQDFYUURXJSL
|
6.1 | Ki | 8 | — | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
RTYJMUXLFRYRBU
|
6.1 | Ki | 35 | — | |
WAKGEHXTOOFEAE
|
6.1 | Ki | 27 | — | |
AAKJLRGGTJKAMG
|
6.0 | Kd | 50 | Yes | |
YYLKKYCXAOBSRM
|
6.0 | Kd | 191 | — | |
DPEXRCOBPACFOO
|
6.0 | Ki | 36 | — | |
FHIVNWJIENRJBH
|
6.0 | Ki | 9 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JHYHWHUTTXJICB
|
6.0 | Ki | 18 | — | |
JMIIFJIJWDCOEP
|
6.0 | Ki | 15 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
SEZFNTZQMWJIAI
|
6.0 | Ki | 22 | — | |
XTVULKIROSNNTG
|
6.0 | Ki | 29 | — | |
XXJWYDDUDKYVKI
|
6.0 | Ki | 52 | — | |
ZHNDVKCPJRLARD
|
6.0 | Ki | 3 | — |