Target Details
| UniProt AC | P29376 |
|---|---|
| Gene Symbol | LTK |
| Protein Name | Leukocyte tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 127
- Clinical molecules 16
- Avg pChEMBL 7.0
Active Molecules (127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GNLAGGCSJGJECE
|
7.1 | Ki | 19 | Yes | |
PROLIXHVRCJEFH
|
7.1 | Ki | 46 | — | |
VCFDMLBPASGZTP
|
7.1 | Ki | 38 | — | |
ZGDYBJXDIXVTLV
|
7.1 | Ki | 54 | — | |
ATGVCJYHNOSZEV
|
7.0 | Ki | 23 | — | |
CXQHYVUVSFXTMY
|
7.0 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.0 | Kd | 149 | — | |
QXIOZIFTPMAING
|
6.9 | IC50 | 17 | — | |
NWMPVMMGSHXANZ
|
6.9 | Ki | 58 | — | |
UIRCQOKSJDLYBB
|
6.9 | Ki | 50 | — | |
WDARYLSSWBWVCU
|
6.9 | Ki | 49 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
NVRXTLZYXZNATH
|
6.8 | Ki | 47 | Yes | |
ODPGGGTTYSGTGO
|
6.8 | Kd | 153 | — | |
QVNZKVACBBTKSL
|
6.8 | Ki | 38 | — | |
NXSJMRCTGYTSTK
|
6.7 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
6.7 | Kd | 170 | — | |
HXHAJRMTJXHJJZ
|
6.7 | Ki | 52 | Yes | |
LUPCHAFIKZSOOK
|
6.7 | Ki | 15 | — | |
VSVWQTDDGQSGHP
|
6.7 | Ki | 51 | — | |
FUMCKNCUEAQHCV
|
6.6 | Ki | 103 | — | |
KUNZDWIFPOMUOX
|
6.6 | Ki | 36 | — | |
ZCCJKVBTHCOISJ
|
6.6 | Ki | 46 | — | |
WVXNSAVVKYZVOE
|
6.6 | IC50 | 92 | — | |
GCDSDVNITVBCDW
|
6.5 | IC50 | 17 | — | |
AUDNGNGLLRZLDR
|
6.5 | Ki | 33 | — | |
JNXJKTXDSPWNRP
|
6.5 | Ki | 30 | — | |
JOGKUKXHTYWRGZ
|
6.5 | Ki | 28 | — | |
MZDKLVOWGIOKTN
|
6.5 | Ki | 80 | — | |
UJBJWYNPUOLFIZ
|
6.4 | IC50 | 49 | — | |
AYXVSCVVQIADBF
|
6.4 | Ki | 10 | — | |
DWTNLZZEPSCAIH
|
6.4 | Ki | 25 | — | |
IFPPYSWJNWHOLQ
|
6.4 | Ki | 52 | Yes | |
OGNYUTNQZVRGMN
|
6.4 | Ki | 16 | Yes | |
RUPJOKGREQMQSI
|
6.4 | Ki | 9 | — | |
VWACUNWBMWWMPJ
|
6.4 | Ki | 18 | — | |
WUTNLCUQZGDRGX
|
6.4 | Ki | 5 | — | |
ZLHFILGSQDJULK
|
6.4 | Ki | 37 | Yes | |
HFNKQEVNSGCOJV
|
6.4 | Kd | 65 | — | |
UIARLYUEJFELEN
|
6.3 | Kd | 289 | Yes | |
GCIKSSRWRFVXBI
|
6.3 | Ki | 109 | Yes | |
JJGSOVIZOMZMCS
|
6.3 | Ki | 35 | — | |
MCKPYPWHBUXLEZ
|
6.3 | Ki | 21 | — | |
MHWHPWMWKYXCRJ
|
6.3 | Ki | 32 | — | |
MMFBBQQGBVPLQQ
|
6.3 | Ki | 13 | — | |
NKEUPUJTVALZIK
|
6.3 | Ki | 28 | — | |
QCOULMVHIHJKFY
|
6.3 | Ki | 14 | — | |
XUFLBSMTYMFOQH
|
6.3 | Ki | 43 | — | |
XZWVOUQIYLZUCJ
|
6.3 | Ki | 23 | — | |
MPVGZUGXCQEXTM
|
6.3 | Kd | 61 | Yes |