Target Details
| UniProt AC | P29376 |
|---|---|
| Gene Symbol | LTK |
| Protein Name | Leukocyte tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 127
- Clinical molecules 16
- Avg pChEMBL 7.0
Active Molecules (127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IUWWRSQCDUQDEZ
|
9.2 | IC50 | 8 | — | |
IUWWRSQCDUQDEZ
|
9.2 | IC50 | 9 | — | |
QQWUGDVOUVUTOY
|
9.0 | Kd | 231 | Yes | |
HZTYDQRUAWIZRE
|
9.0 | Kd | 40 | Yes | |
HAYYBYPASCDWEQ
|
8.8 | Ki | 47 | — | |
WHVFDYQCAMPLMS
|
8.8 | Ki | 20 | Yes | |
DIXMBHMNEHPFCX
|
8.7 | IC50 | 12 | — | |
DLWMVUDMPMKGEE
|
8.7 | Ki | 24 | — | |
WSTUJEXAPHIEIM
|
8.6 | Kd | 10 | — | |
IIXWYSCJSQVBQM
|
8.6 | IC50 | 18 | — | |
VXYZCOCRVAQWBG
|
8.6 | IC50 | 15 | — | |
HKSZLNNOFSGOKW
|
8.5 | Ki | 118 | — | |
OWRXHGAFWZFFCW
|
8.5 | Ki | 113 | — | |
GDRLJBDXWDATLA
|
8.4 | IC50 | 13 | — | |
SDBOIBYRBWPIEL
|
8.4 | Ki | 31 | — | |
LOONVQWRKJLEEG
|
8.2 | IC50 | 8 | — | |
UYJNQQDJUOUFQJ
|
8.1 | Ki | 68 | — | |
GZYCQQBRSRIFII
|
8.1 | Kd | 7 | — | |
JZTOUVBEZONDKA
|
8.0 | Ki | 80 | — | |
LJKJYKWDLJUZHA
|
8.0 | Ki | 24 | — | |
KTEIFNKAUNYNJU
|
8.0 | Ki | 48 | — | |
KTEIFNKAUNYNJU
|
7.9 | Kd | 114 | — | |
DSSRVQAIWBZWON
|
7.9 | Ki | 9 | — | |
HZPACYSNLOCDLW
|
7.9 | Ki | 48 | — | |
AILRADAXUVEEIR
|
7.8 | IC50 | 75 | — | |
RGNHKJWHFIPHIM
|
7.7 | Ki | 66 | — | |
VKBFHTIUXUCYRQ
|
7.7 | Ki | 66 | — | |
VNDWQCSOSCCWIP
|
7.6 | Ki | 39 | Yes | |
NMJMRSQTDLRCRQ
|
7.5 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
7.5 | IC50 | 408 | — | |
ADLPKFFMGIJZIM
|
7.5 | Ki | 44 | — | |
LBVKEEFIPBQIMD
|
7.5 | Ki | 27 | — | |
XKFTZKGMDDZMJI
|
7.5 | Ki | 56 | — | |
RYYNGWLOYLRZLK
|
7.4 | Ki | 104 | — | |
WPHKIQPVPYJNAX
|
7.4 | Ki | 81 | — | |
VWCZORWQNKCYGE
|
7.4 | IC50 | 17 | — | |
UMBIRSZUCJNBHB
|
7.3 | IC50 | 18 | — | |
HDRLAVNNWSHSOA
|
7.3 | Ki | 19 | — | |
ORRHVRJUSPCILV
|
7.3 | Ki | 16 | — | |
QLWUDWMYFSWGHK
|
7.3 | Ki | 22 | — | |
GLDSKRNGVVYJAB
|
7.3 | Kd | 16 | — | |
SGZZQKMOFHIDKW
|
7.3 | Kd | 13 | — | |
HFNKQEVNSGCOJV
|
7.2 | Ki | 18 | — | |
MGGBYMDAPCCKCT
|
7.2 | IC50 | 23 | — | |
GJKVMXDBPDDFHI
|
7.2 | Ki | 27 | — | |
XJSFDMGICAWQFS
|
7.2 | Ki | 60 | — | |
JOAFWIHZEBKYQK
|
7.2 | IC50 | 10 | — | |
ROHJEIACUNTGFP
|
7.2 | IC50 | 16 | — | |
AEYLJTAIDDIOBA
|
7.1 | Ki | 53 | — | |
BRTHUECZMVKNMQ
|
7.1 | Ki | 31 | — |