Target Details
| UniProt AC | P29375 |
|---|---|
| Gene Symbol | KDM5A |
| Protein Name | Lysine-specific demethylase 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 240
- Clinical molecules 0
- Avg pChEMBL 6.55
Associated Diseases (1)
Active Molecules (240)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MBJOZIBNEMTKKO
|
6.0 | IC50 | 3 | — | |
MBWGIVXATSPGAT
|
6.0 | IC50 | 3 | — | |
MDBCUBGXHYXSNR
|
6.0 | IC50 | 2 | — | |
MKZLVNIZKIFRHO
|
6.0 | IC50 | 3 | — | |
MVDDWOUDRGQZND
|
6.0 | IC50 | 2 | — | |
MWJQMQXBUJYTHO
|
6.0 | IC50 | 4 | — | |
NBKPXVZLKABEHX
|
6.0 | IC50 | 3 | — | |
NCASPJRQDUQONI
|
6.0 | IC50 | 3 | — | |
NUKWFAQUBJIRPU
|
6.0 | IC50 | 3 | — | |
NZRXUQUWPPLOHA
|
6.0 | IC50 | 3 | — | |
OJXCGLCDLOSZJU
|
6.0 | IC50 | 2 | — | |
ONKWECDQZPASOC
|
6.0 | IC50 | 4 | — | |
PVQPINFUKHIDOU
|
6.0 | IC50 | 3 | — | |
PXPKNVPANSVBHA
|
6.0 | IC50 | 3 | — | |
QNCYOEYMNMZNBO
|
6.0 | IC50 | 3 | — | |
RABORKCQNWSDEB
|
6.0 | IC50 | 2 | — | |
RYHMPYHFLUZIAQ
|
6.0 | IC50 | 3 | — | |
SGSDGKOZKXKUJL
|
6.0 | IC50 | 2 | — | |
SSRPMNPULVBKPU
|
6.0 | IC50 | 2 | — | |
TVOKPAHWCXXTHY
|
6.0 | IC50 | 3 | — | |
TYQVGBHPIVDCJP
|
6.0 | IC50 | 4 | — | |
UEFZTBOXYTUEQA
|
6.0 | IC50 | 4 | — | |
UMHHZTUSDDYOHB
|
6.0 | IC50 | 2 | — | |
UQVSSWJZBFXFEN
|
6.0 | IC50 | 3 | — | |
VFQWDEDHEXEJLC
|
6.0 | IC50 | 3 | — | |
VMLMHVMQZCMCBR
|
6.0 | IC50 | 4 | — | |
VTUTUCVVSXMISL
|
6.0 | IC50 | 3 | — | |
WGDUIIXPWPBNOF
|
6.0 | IC50 | 3 | — | |
WJNMKYLJNLYALB
|
6.0 | IC50 | 4 | — | |
XFBUWKQDOAULCT
|
6.0 | IC50 | 3 | — | |
XSSUXYYELFOOBB
|
6.0 | IC50 | 3 | — | |
YALQAUZSXADMLL
|
6.0 | IC50 | 3 | — | |
YEIUTPICFPHMSZ
|
6.0 | IC50 | 4 | — | |
YHNFXISQPODBJA
|
6.0 | IC50 | 2 | — | |
YMTUVGRFKLITAS
|
6.0 | IC50 | 3 | — | |
YMWREFXLGWZZOR
|
6.0 | IC50 | 5 | — | |
YOZDGVQEWQPZKP
|
6.0 | IC50 | 2 | — | |
YVPHKAZMKGNDEA
|
6.0 | IC50 | 2 | — | |
YYOBYQZCYKMCFA
|
6.0 | IC50 | 4 | — | |
ZQVGHRRKWOITDJ
|
6.0 | IC50 | 4 | — |