Target Details
| UniProt AC | P29375 |
|---|---|
| Gene Symbol | KDM5A |
| Protein Name | Lysine-specific demethylase 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 240
- Clinical molecules 0
- Avg pChEMBL 6.55
Associated Diseases (1)
Active Molecules (240)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QKDWURZWFKZKLH
|
6.3 | IC50 | 3 | — | |
QUEUBIKJDGXLFY
|
6.3 | IC50 | 3 | — | |
QVSDPEWGBYKEDU
|
6.3 | IC50 | 4 | — | |
RCFPZNIWZQNDJL
|
6.3 | IC50 | 3 | — | |
REFIQVNXDXIMLX
|
6.3 | IC50 | 3 | — | |
RFGNJZHABKKPLK
|
6.3 | IC50 | 2 | — | |
RMCMBFPHTFWEBT
|
6.3 | IC50 | 2 | — | |
RNHDGJROFDMRJA
|
6.3 | IC50 | 3 | — | |
RPOONZXSYGAYQG
|
6.3 | IC50 | 3 | — | |
SEHBCCOGWMQNBD
|
6.3 | IC50 | 3 | — | |
SIFAONGGESBNMT
|
6.3 | IC50 | 2 | — | |
TUXVCHDESZTZON
|
6.3 | IC50 | 2 | — | |
UDNZKYWBVTTWJF
|
6.3 | IC50 | 5 | — | |
UFXLKZLYQGPHTG
|
6.3 | IC50 | 3 | — | |
UNPSHKPWHBDUJV
|
6.3 | IC50 | 2 | — | |
UQZWANPYQUOQKJ
|
6.3 | IC50 | 3 | — | |
VESNHHASMCDWDO
|
6.3 | IC50 | 3 | — | |
VYUQZEXRXAXQKG
|
6.3 | IC50 | 4 | — | |
WBNKZKXRLUOOMX
|
6.3 | IC50 | 3 | — | |
WTMJZFIQFSYVHA
|
6.3 | IC50 | 4 | — | |
WTVJIZOUDVEZFE
|
6.3 | IC50 | 3 | — | |
WVEHUIVVPBXOJC
|
6.3 | IC50 | 5 | — | |
WXKUUFVPZNAMJQ
|
6.3 | IC50 | 3 | — | |
XEOWFNYWWSWLBN
|
6.3 | IC50 | 3 | — | |
XGBOARWPNSLLHZ
|
6.3 | IC50 | 4 | — | |
XRHOGEKRJFLZGA
|
6.3 | IC50 | 3 | — | |
XUYSGGCAQKHJKY
|
6.3 | IC50 | 2 | — | |
XYHXZRBZNBOLAJ
|
6.3 | IC50 | 3 | — | |
YCGATGBJHALDLT
|
6.3 | IC50 | 3 | — | |
YWMPCCYNGABIMS
|
6.3 | IC50 | 4 | — | |
ZPFAMOBPFNYKFI
|
6.3 | IC50 | 3 | — | |
ZTSZMVPLKHSHGA
|
6.3 | IC50 | 3 | — | |
RBGNHCYGFBRIRO
|
6.2 | IC50 | 3 | — | |
MJIVRKPEXXHNJT
|
6.1 | IC50 | 9 | — | |
XTTNXYOVGZYVFK
|
6.1 | IC50 | 2 | — | |
AGEAFYTUQGJREF
|
6.0 | IC50 | 3 | — | |
BBJLCHZEGBSIFB
|
6.0 | IC50 | 2 | — | |
BUWBKFLUJJAMOD
|
6.0 | IC50 | 2 | — | |
CXXOKDSMTHKIAI
|
6.0 | IC50 | 2 | — | |
DBNRSQHWQKIXGR
|
6.0 | IC50 | 3 | — | |
DNNQPECTYYGIPO
|
6.0 | IC50 | 3 | — | |
FISNSBBQGXNIJS
|
6.0 | IC50 | 2 | — | |
FNPHROKMXPECAD
|
6.0 | IC50 | 4 | — | |
FWSGIYDMJPQQGL
|
6.0 | IC50 | 4 | — | |
HWBFUMCZKFJIFB
|
6.0 | IC50 | 3 | — | |
JESVJQKIAGLWLN
|
6.0 | IC50 | 2 | — | |
JFEKVRDZSRWNEZ
|
6.0 | IC50 | 2 | — | |
KGVYZQBMOYMEEW
|
6.0 | IC50 | 2 | — | |
LFTMQFRCMXWVBO
|
6.0 | IC50 | 3 | — | |
LINOVANVVSYFAN
|
6.0 | IC50 | 2 | — |