Target Details
| UniProt AC | P29375 |
|---|---|
| Gene Symbol | KDM5A |
| Protein Name | Lysine-specific demethylase 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 240
- Clinical molecules 0
- Avg pChEMBL 6.55
Associated Diseases (1)
Active Molecules (240)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FRSFPMMQGXIOOY
|
6.3 | IC50 | 3 | — | |
GAAWGDKZMZYRLG
|
6.3 | IC50 | 3 | — | |
GBJNSFXBUOTPIV
|
6.3 | IC50 | 3 | — | |
GLMOOUIHDMOTSN
|
6.3 | IC50 | 3 | — | |
HMFDIJHBCQAEDL
|
6.3 | IC50 | 3 | — | |
HONRHPVMYYIRBL
|
6.3 | IC50 | 3 | — | |
HVUATMMGHIDJOR
|
6.3 | IC50 | 2 | — | |
HYSAXCDPGIPIAF
|
6.3 | IC50 | 3 | — | |
IKDUYJZLUXCOMP
|
6.3 | IC50 | 4 | — | |
IOCMNXRIFNSUHI
|
6.3 | IC50 | 3 | — | |
IWXQPCTUWUKXSM
|
6.3 | IC50 | 2 | — | |
JFUSDWYLUAUIKN
|
6.3 | IC50 | 5 | — | |
JQPYWFPJAZZKAV
|
6.3 | IC50 | 5 | — | |
KAHITAMALHBXDQ
|
6.3 | IC50 | 3 | — | |
KBYPMYYZRUNPRA
|
6.3 | IC50 | 3 | — | |
KLXSSSNBZFSVGC
|
6.3 | IC50 | 3 | — | |
KPJOSXHPFIXXLA
|
6.3 | IC50 | 4 | — | |
LFQKFAJAKGJKJE
|
6.3 | IC50 | 2 | — | |
LJSLTRVLEYBZQF
|
6.3 | IC50 | 2 | — | |
LKBZHRSAENXIOI
|
6.3 | IC50 | 4 | — | |
LLIMXLUTGJVMBY
|
6.3 | IC50 | 4 | — | |
LMWRRFGBEDJAGG
|
6.3 | IC50 | 3 | — | |
LPFWATLXDCIHNH
|
6.3 | IC50 | 2 | — | |
LQNSEJCSWWGGGC
|
6.3 | IC50 | 3 | — | |
MDKIIFAUVUDOPJ
|
6.3 | IC50 | 3 | — | |
MDRIPRQWTFFXTF
|
6.3 | IC50 | 3 | — | |
MFXLJRSRCQXMLR
|
6.3 | IC50 | 3 | — | |
MITOFELVTHNBGA
|
6.3 | IC50 | 3 | — | |
MJGNHAKBDPMKTA
|
6.3 | IC50 | 2 | — | |
MMZVVWIDZXOSFA
|
6.3 | IC50 | 3 | — | |
MWBHFQQDMCLDJK
|
6.3 | IC50 | 3 | — | |
MYEIDQDVSWLKKZ
|
6.3 | IC50 | 2 | — | |
MYIZAYXMTDPUHW
|
6.3 | IC50 | 3 | — | |
MYWICJXUGCWVAW
|
6.3 | IC50 | 4 | — | |
NCCRYWGVCKYSTJ
|
6.3 | IC50 | 3 | — | |
NFVXMQNDOGMBRE
|
6.3 | IC50 | 3 | — | |
NRGSAZMZQWJSRB
|
6.3 | IC50 | 3 | — | |
NUHPPDIXDWJTCM
|
6.3 | IC50 | 3 | — | |
OAVHESBEECDWSL
|
6.3 | IC50 | 2 | — | |
OKWTXEOPPSGVKX
|
6.3 | IC50 | 2 | — | |
OTBZGJHFGXDSHF
|
6.3 | IC50 | 4 | — | |
OWZXJIAEISCANW
|
6.3 | IC50 | 3 | — | |
OYXGRLHUDVMFKK
|
6.3 | IC50 | 3 | — | |
PPJJPXKKNDUAAE
|
6.3 | IC50 | 3 | — | |
QBJBXNHYPDLIAQ
|
6.3 | IC50 | 2 | — | |
QBLUFCRSMWHQNN
|
6.3 | IC50 | 3 | — | |
QFWIUYKPWXTXGH
|
6.3 | IC50 | 2 | — | |
QGEQDCNJTLKLCD
|
6.3 | IC50 | 3 | — | |
QGWDKDJPSMMAIM
|
6.3 | IC50 | 2 | — | |
QKDSOTUHFJKBQW
|
6.3 | IC50 | 3 | — |