Target Details
| UniProt AC | P29375 |
|---|---|
| Gene Symbol | KDM5A |
| Protein Name | Lysine-specific demethylase 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 240
- Clinical molecules 0
- Avg pChEMBL 6.55
Associated Diseases (1)
Active Molecules (240)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GMWKOCOYZWNSIJ
|
7.0 | IC50 | 3 | — | |
ICHXMUXDEGLEPY
|
7.0 | IC50 | 2 | — | |
JHDVDMCSBXSGFG
|
7.0 | IC50 | 3 | — | |
JYEUQFOUZAUNTD
|
7.0 | IC50 | 2 | — | |
LJHFNRZRNINLGH
|
7.0 | IC50 | 3 | — | |
NHSZAIFDCXEIFA
|
7.0 | IC50 | 3 | — | |
RHPSPIUSPOTEGT
|
7.0 | IC50 | 2 | — | |
SMXDPQZYSIFABV
|
7.0 | IC50 | 3 | — | |
WAPIESSEOAYVNJ
|
7.0 | IC50 | 5 | — | |
WBQBJTNMBDYBHL
|
7.0 | IC50 | 3 | — | |
WPESTWIANQBENM
|
7.0 | IC50 | 2 | — | |
YFUUKCJIHIACCK
|
7.0 | IC50 | 3 | — | |
YTKUKFQCCYBMFH
|
7.0 | IC50 | 2 | — | |
ZMBZYRJHWCFIQA
|
7.0 | IC50 | 2 | — | |
ZNABVSMDKOBVOS
|
7.0 | IC50 | 3 | — | |
ZQNXWEZQRNBWCU
|
7.0 | IC50 | 5 | — | |
OEHJHVSOQQJIGN
|
6.7 | IC50 | 3 | — | |
OXELDRCVUWWSFZ
|
6.7 | IC50 | 3 | — | |
SPGCFZXNJYGZNU
|
6.6 | IC50 | 2 | — | |
YHHFKWKMXWRVTJ
|
6.6 | IC50 | 7 | — | |
YSLNSTXNXMRWMU
|
6.6 | IC50 | 3 | — | |
VICDONOMNXVSDL
|
6.6 | IC50 | 2 | — | |
VHKSSHRSJGZQOV
|
6.5 | IC50 | 4 | — | |
WCILOMUUNVPIKQ
|
6.5 | IC50 | 5 | — | |
WXFDDWMINUVYFL
|
6.5 | IC50 | 4 | — | |
PATSJMHSNAENAO
|
6.5 | IC50 | 2 | — | |
NIROIUUITQXVHP
|
6.5 | IC50 | 2 | — | |
BGMIWCIVXVXHDU
|
6.5 | IC50 | 3 | — | |
RVWFSGMSJSTAIJ
|
6.4 | IC50 | 2 | — | |
ABANEZXFVFHRMY
|
6.3 | IC50 | 2 | — | |
BEOSCPUYUHDKBT
|
6.3 | IC50 | 3 | — | |
BNEDYWDXODJLAY
|
6.3 | IC50 | 5 | — | |
BVUXJIUJKSADTM
|
6.3 | IC50 | 3 | — | |
CBVFSACWQSKTBS
|
6.3 | IC50 | 2 | — | |
CDCAKPHONNAIQI
|
6.3 | IC50 | 2 | — | |
CXAIXDFFEAKNFB
|
6.3 | IC50 | 3 | — | |
DADJCXBYNKOCQO
|
6.3 | IC50 | 3 | — | |
DEOQWVFWHCSFQH
|
6.3 | IC50 | 3 | — | |
DGPKTIKFLWFZTL
|
6.3 | IC50 | 3 | — | |
DGPKTIKFLWFZTL
|
6.3 | IC50 | 3 | — | |
DJOUORRZKJVHJG
|
6.3 | IC50 | 2 | — | |
DQZXWCVKIBSQAJ
|
6.3 | IC50 | 3 | — | |
DRXNXOKZAZEGFK
|
6.3 | IC50 | 3 | — | |
DTJUHOKYRUAGQQ
|
6.3 | IC50 | 3 | — | |
DYVKRSMFVROHFY
|
6.3 | IC50 | 2 | — | |
FEZIKLVLFANZBD
|
6.3 | IC50 | 4 | — | |
FJDQJUPBHKHILS
|
6.3 | IC50 | 4 | — | |
FODSHMOMERZNFO
|
6.3 | IC50 | 2 | — | |
FPJJSKKWGRACAX
|
6.3 | IC50 | 3 | — | |
FQGUTBFYFQAJJX
|
6.3 | IC50 | 2 | — |