Target Details
UniProt ACP29375
Gene SymbolKDM5A
Protein NameLysine-specific demethylase 5A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2)
Summary
  • Multi-target molecules 240
  • Clinical molecules 0
  • Avg pChEMBL 6.55
Top Co-occurrence Targets
Active Molecules (240)
InChIKey pChEMBL Type Targets Clinical
ZVDVVBQKFXBYJN 8.9 IC50 4
ALHWXWTUDYISRS 8.5 IC50 3
WVXRMWSXRNMWLL 8.4 IC50 4
MZLRXFKOAWCNNY 8.4 IC50 3
ITIAJFABKUNVBR 8.2 IC50 2
TUVMHEGGYLIJHD 8.0 IC50 3
LNMSTPSCCSYARO 7.9 IC50 2
TVFQMRCHDYLPNH 7.9 IC50 3
PSOBPHXKKHPWMU 7.9 IC50 10
HJFUZTRJZDWWPG 7.8 IC50 2
NKHXMCLESKPQJD 7.8 IC50 3
BFUDSGXVTFJZFS 7.8 IC50 2
KRXWJZIHQRIGSJ 7.8 IC50 3
VAHFPFWYMCULAM 7.8 IC50 2
DOZDKMPUJLMVHD 7.7 IC50 2
UTLFDRFGHDOZAU 7.7 IC50 2
GTWJZXSSCNHGGN 7.7 IC50 3
AEGZTINJBDVGEP 7.7 IC50 2
DHXKRMSKXLDZGY 7.7 IC50 3
LGZJVCBTCCGZTI 7.7 IC50 2
QFOYPGLCAPECCY 7.7 IC50 2
HJWSLDFYCQJXLZ 7.6 IC50 3
UHVUUCAAVHIPKM 7.6 IC50 2
ZTYRLXUTLYBVHH 7.6 IC50 8
BJPPOTJAQZGVIA 7.6 IC50 4
NPAMRWDIMURYSE 7.6 IC50 3
RGGMVQDDHDCRDM 7.6 IC50 9
WBWADLLKNGUCBS 7.6 IC50 2
MEUCYOUPEAATQR 7.6 IC50 2
QZXMTFZQLZHLTN 7.5 IC50 3
CEGMXGCEQZMHBD 7.5 IC50 3
NNMOCDJHJWOBLY 7.5 IC50 4
OAJKLLSETTZMPH 7.5 IC50 3
ROLKCSJSIFETFK 7.5 IC50 3
NYJLXELRMWJXFN 7.4 IC50 3
ZQSAQSCGHSOXTE 7.4 IC50 2
MKBWAOCGFREQKS 7.4 IC50 4
CXEXTVGTDZRKJS 7.3 IC50 3
AMVDOFFKSJJORQ 7.3 IC50 2
NGZUHYKCIFSOED 7.3 IC50 3
XHLDZZFRSRZGNZ 7.3 IC50 3
QVELLOOBNULIGQ 7.2 IC50 3
DSGOLESVOJUGOK 7.2 IC50 4
PNFMVADNCOGWME 7.2 IC50 4
CCXBVLGMHSEBLX 7.1 IC50 4
QUWILIWFYYFAPG 7.1 IC50 3
MAYCQAAYKTWJKJ 7.1 IC50 3
WNSMPEBHTSITSG 7.1 IC50 3
BJFOUULYELAMPD 7.0 IC50 3
CDSIWRGJSKHJRV 7.0 IC50 2
2D structure