Target Details
| UniProt AC | P29375 |
|---|---|
| Gene Symbol | KDM5A |
| Protein Name | Lysine-specific demethylase 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 240
- Clinical molecules 0
- Avg pChEMBL 6.55
Associated Diseases (1)
Active Molecules (240)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZVDVVBQKFXBYJN
|
8.9 | IC50 | 4 | — | |
ALHWXWTUDYISRS
|
8.5 | IC50 | 3 | — | |
WVXRMWSXRNMWLL
|
8.4 | IC50 | 4 | — | |
MZLRXFKOAWCNNY
|
8.4 | IC50 | 3 | — | |
ITIAJFABKUNVBR
|
8.2 | IC50 | 2 | — | |
TUVMHEGGYLIJHD
|
8.0 | IC50 | 3 | — | |
LNMSTPSCCSYARO
|
7.9 | IC50 | 2 | — | |
TVFQMRCHDYLPNH
|
7.9 | IC50 | 3 | — | |
PSOBPHXKKHPWMU
|
7.9 | IC50 | 10 | — | |
HJFUZTRJZDWWPG
|
7.8 | IC50 | 2 | — | |
NKHXMCLESKPQJD
|
7.8 | IC50 | 3 | — | |
BFUDSGXVTFJZFS
|
7.8 | IC50 | 2 | — | |
KRXWJZIHQRIGSJ
|
7.8 | IC50 | 3 | — | |
VAHFPFWYMCULAM
|
7.8 | IC50 | 2 | — | |
DOZDKMPUJLMVHD
|
7.7 | IC50 | 2 | — | |
UTLFDRFGHDOZAU
|
7.7 | IC50 | 2 | — | |
GTWJZXSSCNHGGN
|
7.7 | IC50 | 3 | — | |
AEGZTINJBDVGEP
|
7.7 | IC50 | 2 | — | |
DHXKRMSKXLDZGY
|
7.7 | IC50 | 3 | — | |
LGZJVCBTCCGZTI
|
7.7 | IC50 | 2 | — | |
QFOYPGLCAPECCY
|
7.7 | IC50 | 2 | — | |
HJWSLDFYCQJXLZ
|
7.6 | IC50 | 3 | — | |
UHVUUCAAVHIPKM
|
7.6 | IC50 | 2 | — | |
ZTYRLXUTLYBVHH
|
7.6 | IC50 | 8 | — | |
BJPPOTJAQZGVIA
|
7.6 | IC50 | 4 | — | |
NPAMRWDIMURYSE
|
7.6 | IC50 | 3 | — | |
RGGMVQDDHDCRDM
|
7.6 | IC50 | 9 | — | |
WBWADLLKNGUCBS
|
7.6 | IC50 | 2 | — | |
MEUCYOUPEAATQR
|
7.6 | IC50 | 2 | — | |
QZXMTFZQLZHLTN
|
7.5 | IC50 | 3 | — | |
CEGMXGCEQZMHBD
|
7.5 | IC50 | 3 | — | |
NNMOCDJHJWOBLY
|
7.5 | IC50 | 4 | — | |
OAJKLLSETTZMPH
|
7.5 | IC50 | 3 | — | |
ROLKCSJSIFETFK
|
7.5 | IC50 | 3 | — | |
NYJLXELRMWJXFN
|
7.4 | IC50 | 3 | — | |
ZQSAQSCGHSOXTE
|
7.4 | IC50 | 2 | — | |
MKBWAOCGFREQKS
|
7.4 | IC50 | 4 | — | |
CXEXTVGTDZRKJS
|
7.3 | IC50 | 3 | — | |
AMVDOFFKSJJORQ
|
7.3 | IC50 | 2 | — | |
NGZUHYKCIFSOED
|
7.3 | IC50 | 3 | — | |
XHLDZZFRSRZGNZ
|
7.3 | IC50 | 3 | — | |
QVELLOOBNULIGQ
|
7.2 | IC50 | 3 | — | |
DSGOLESVOJUGOK
|
7.2 | IC50 | 4 | — | |
PNFMVADNCOGWME
|
7.2 | IC50 | 4 | — | |
CCXBVLGMHSEBLX
|
7.1 | IC50 | 4 | — | |
QUWILIWFYYFAPG
|
7.1 | IC50 | 3 | — | |
MAYCQAAYKTWJKJ
|
7.1 | IC50 | 3 | — | |
WNSMPEBHTSITSG
|
7.1 | IC50 | 3 | — | |
BJFOUULYELAMPD
|
7.0 | IC50 | 3 | — | |
CDSIWRGJSKHJRV
|
7.0 | IC50 | 2 | — |