Target Details
UniProt ACP29371
Gene SymbolTACR3
Protein NameNeuromedin-K receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 164
  • Clinical molecules 0
  • Avg pChEMBL 7.92
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (164)
InChIKey pChEMBL Type Targets Clinical
FLNYCRJBCNNHRH 8.6 Ki 3
LWENKLDZCHEYBQ 8.6 Kd 2
GXKBHFYZTAQYCX 8.6 Ki 2
MUZRICFSRACWJI 8.6 IC50 3
HGZMZNGGJOZVFE 8.5 Ki 2
QOOXCQFWUYVSGU 8.5 Ki 2
JMEKLKBPAWJBOV 8.5 Ki 3
HNYCTUJIKKNHPR 8.5 Ki 3
GGXDLXDHGKHOEN 8.5 Ki 2
SUCQKPUTZDUCKO 8.5 Ki 3
KQNYTTDHCMFOME 8.5 IC50 2
BIAVGWDGIJKWRM 8.4 Ki 2
KGORHDRKRVOPJF 8.3 Ki 2
UZIUERPVGXNKKW 8.3 Ki 3
KIWPQCODGUAEAZ 8.3 Ki 2
RVDBXUCLTPUWIX 8.3 Ki 2
VPPFVSVLCATXPY 8.3 Ki 2
MQNYRKWJSMQECI 8.3 Ki 2
HJXINJBZYGSKKL 8.2 IC50 2
DGLDUQZIRFLLRH 8.2 Ki 3
ZSIQAOCNFRWDNJ 8.2 IC50 2
ZXJRUKOAFOUFIR 8.2 Ki 2
HPPQGIFLKZFURI 8.2 IC50 3
MQNYRKWJSMQECI 8.2 IC50 2
CYDMWSSMUBQXRD 8.2 Ki 2
MHEYENUCWKQKPB 8.2 Ki 2
XDFFVHQCALIXPH 8.1 Ki 2
JEZKKPXWSVQUPH 8.1 Ki 3
OFXGPUCSXYQAEH 8.1 Ki 2
IOIJNSLWZAOUPA 8.1 Ki 2
ODPRNYGWGVRXIG 8.1 IC50 3
QBFWYYRMUQGGNR 8.1 Ki 2
XAQPCKKFCKSQOW 8.1 IC50 2
KYIGOCCCBXRHNJ 8.1 IC50 43
CYDMWSSMUBQXRD 8.1 Ki 2
OJNYEFLQZAKWEW 8.0 Ki 3
NHXYSAFTNPANFK 8.0 IC50 3
ZZFJEAWXKJAJIS 8.0 Ki 3
OZJDKUMSRQSURZ 8.0 Ki 3
FRDDXKUSVLZWRL 8.0 Ki 3
OFUFYXNPWNFQBY 8.0 Ki 3
XCCMZNKLKPVPJT 8.0 IC50 2
DGDAEJXIYKFTSC 7.9 Kd 2
NFUWMFTULXHEKZ 7.9 Ki 2
VMUJISIYYNPJBE 7.9 Ki 3
VVRKQCXRSANSIV 7.9 Ki 2
MXNGYQJJYRVGGJ 7.9 Ki 2
MSGGUBXMXWEJRT 7.8 Ki 2
HCGIROBRNBTDFG 7.8 Kd 2
YSDZQWRVRDWYHN 7.8 IC50 2
2D structure