Target Details
| UniProt AC | P29350 |
|---|---|
| Gene Symbol | PTPN6 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00017 (SH2) PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 6.39
KEGG Pathways (11)
- Adherens junction
- B cell receptor signaling pathway
- Efferocytosis
- IgSF CAM signaling
- JAK-STAT signaling pathway
- Leishmaniasis
- Natural killer cell mediated cytotoxicity
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathogenic Escherichia coli infection
- Proteoglycans in cancer
- T cell receptor signaling pathway
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZNUFCVFEZWEKRQ
|
7.0 | IC50 | 2 | — | |
CQHDXEWKDCKMHF
|
6.9 | IC50 | 6 | — | |
RNFXSRZAAHHCDB
|
6.7 | IC50 | 2 | — | |
LVGFRMIIXODOEQ
|
6.5 | IC50 | 4 | — | |
SFPAQPMKUYAZGZ
|
6.4 | IC50 | 3 | — | |
XKVWTVIOHRIVIZ
|
6.4 | IC50 | 4 | — | |
BEWNGQMBEVZWOA
|
6.3 | IC50 | 4 | — | |
IBIICFQQAQDOQU
|
6.2 | IC50 | 3 | — | |
WVNQJOXFTBTXOE
|
6.1 | IC50 | 6 | — | |
SHUIZLANTVXOQC
|
6.1 | IC50 | 3 | — | |
OBQZFTRIINNEEB
|
6.0 | IC50 | 3 | — | |
ZAKVHDWXAFAMTH
|
6.0 | IC50 | 8 | — |