Target Details
| UniProt AC | P29323 |
|---|---|
| Gene Symbol | EPHB2 |
| Protein Name | Ephrin type-B receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 43
- Clinical molecules 9
- Avg pChEMBL 7.13
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (43)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTWMOWRMSZZHDR
|
8.9 | IC50 | 13 | — | |
AQSSMEORRLJZLU
|
8.7 | Kd | 34 | Yes | |
ZCCPLJOKGAACRT
|
8.6 | IC50 | 599 | — | |
ZBNZXTGUTAYRHI
|
8.6 | Kd | 102 | Yes | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
CXQHYVUVSFXTMY
|
8.4 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
SFCBIFOAGRZJNX
|
8.2 | Kd | 22 | — | |
UBPYILGKFZZVDX
|
8.1 | Kd | 130 | Yes | |
LQSGDXCDNZWTJN
|
8.0 | IC50 | 17 | — | |
VAARYSWULJUGST
|
7.7 | Kd | 119 | Yes | |
SPMVMDHWKHCIDT
|
7.6 | IC50 | 30 | — | |
BNRXMSGHPVYSDK
|
7.6 | IC50 | 24 | — | |
MIMOHMCANSGXIG
|
7.6 | IC50 | 15 | — | |
SPMVMDHWKHCIDT
|
7.6 | IC50 | 5 | — | |
YHVHYWYQEFELOW
|
7.5 | IC50 | 44 | — | |
UEFCSGDOOJJXTN
|
7.4 | IC50 | 46 | — | |
QTFCKBFCXDAZIU
|
7.3 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.2 | Kd | 64 | Yes | |
AIKGYQDFIJRQIY
|
7.2 | IC50 | 9 | — | |
UMBFDGUGXMOMHX
|
7.1 | IC50 | 12 | — | |
ZJQYVSTVRXOFQL
|
7.1 | IC50 | 4 | — | |
PCSKFQHKWWNIKM
|
7.0 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
6.9 | IC50 | 408 | — | |
ODPGGGTTYSGTGO
|
6.9 | Kd | 153 | — | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
IUGBGEUCXVKGQK
|
6.6 | Kd | 13 | — | |
UQRCJCNVNUFYDX
|
6.5 | Kd | 27 | — | |
WVXNSAVVKYZVOE
|
6.5 | IC50 | 92 | — | |
MVCOAUNKQVWQHZ
|
6.4 | Kd | 54 | Yes | |
UHTHHESEBZOYNR
|
6.4 | Kd | 66 | Yes | |
HVXKQKFEHMGHSL
|
6.3 | Kd | 21 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes | |
MWKSRKSEWLRPBL
|
6.2 | IC50 | 1075 | — | |
HHZIURLSWUIHRB
|
6.2 | Kd | 57 | Yes | |
SMPGEBOIKULBCT
|
6.2 | IC50 | 15 | — | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
DJYWRQSMWCFDQX
|
6.1 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
NXSJMRCTGYTSTK
|
6.0 | Kd | 200 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |