Target Details
| UniProt AC | P29322 |
|---|---|
| Gene Symbol | EPHA8 |
| Protein Name | Ephrin type-A receptor 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 33
- Clinical molecules 13
- Avg pChEMBL 7.12
KEGG Pathways (1)
Active Molecules (33)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
9.6 | Kd | 102 | Yes | |
ZCCPLJOKGAACRT
|
8.9 | IC50 | 599 | — | |
CXQHYVUVSFXTMY
|
8.7 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
8.7 | Kd | 149 | — | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
JTWMOWRMSZZHDR
|
8.3 | IC50 | 13 | — | |
VAARYSWULJUGST
|
8.2 | Kd | 119 | Yes | |
UBPYILGKFZZVDX
|
8.1 | Kd | 130 | Yes | |
ODPGGGTTYSGTGO
|
7.7 | Kd | 153 | — | |
QNABDSWBQJKBHK
|
7.7 | IC50 | 45 | — | |
UEFCSGDOOJJXTN
|
7.5 | IC50 | 46 | — | |
HHZIURLSWUIHRB
|
7.4 | Kd | 57 | Yes | |
IUGBGEUCXVKGQK
|
7.1 | Kd | 13 | — | |
UHTHHESEBZOYNR
|
7.0 | Kd | 66 | Yes | |
DSZLKOXKYRREEO
|
7.0 | IC50 | 10 | — | |
HKSZLNNOFSGOKW
|
6.7 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.7 | Kd | 213 | — | |
MWKSRKSEWLRPBL
|
6.7 | IC50 | 1075 | — | |
APPXQUDJLJXULP
|
6.6 | IC50 | 47 | — | |
MFAQYJIYDMLAIM
|
6.6 | Kd | 130 | Yes | |
MVCOAUNKQVWQHZ
|
6.6 | Kd | 54 | Yes | |
KTEIFNKAUNYNJU
|
6.5 | Kd | 114 | — | |
WVUNYSQLFKLYNI
|
6.4 | Kd | 46 | Yes | |
YMSXHRWUGLAAKL
|
6.4 | IC50 | 14 | Yes | |
GCIKSSRWRFVXBI
|
6.3 | Kd | 109 | Yes | |
CMJJZRAAQMUAFH
|
6.3 | Kd | 9 | — | |
VYPGLYMWNDRFGZ
|
6.2 | Kd | 12 | — | |
OMZCMEYTWSXEPZ
|
6.1 | Kd | 43 | Yes | |
AAKJLRGGTJKAMG
|
6.0 | Kd | 50 | Yes | |
MLDQJTXFUGDVEO
|
6.0 | Kd | 85 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |