Target Details
| UniProt AC | P29320 |
|---|---|
| Gene Symbol | EPHA3 |
| Protein Name | Ephrin type-A receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF07647 (SAM_2) |
Summary
- Multi-target molecules 34
- Clinical molecules 9
- Avg pChEMBL 7.4
KEGG Pathways (1)
Active Molecules (34)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
10.0 | Kd | 102 | Yes | |
SFCBIFOAGRZJNX
|
10.0 | Kd | 22 | — | |
ZCCPLJOKGAACRT
|
9.5 | IC50 | 599 | — | |
CXQHYVUVSFXTMY
|
9.0 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
9.0 | Kd | 149 | — | |
SUXYGJZMCWKJJI
|
8.9 | IC50 | 26 | Yes | |
ZCWXCBKGPJOAFQ
|
8.3 | IC50 | 13 | — | |
UBPYILGKFZZVDX
|
8.2 | Kd | 130 | Yes | |
VAARYSWULJUGST
|
8.1 | Kd | 119 | Yes | |
ZHMCGBRGDVCXLS
|
8.1 | Kd | 5 | — | |
LYADGAGFYYXXIO
|
7.7 | IC50 | 82 | — | |
DPSNOZFUMXEANO
|
7.6 | Kd | 7 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
7.5 | IC50 | 408 | — | |
RQXYLZHJULSWPX
|
7.4 | Kd | 2 | — | |
JTWMOWRMSZZHDR
|
7.4 | IC50 | 13 | — | |
GZGRGXPFYDFNHF
|
7.3 | Kd | 3 | — | |
MWKSRKSEWLRPBL
|
7.3 | IC50 | 1075 | — | |
UEFCSGDOOJJXTN
|
7.3 | IC50 | 46 | — | |
ODPGGGTTYSGTGO
|
7.1 | Kd | 153 | — | |
HHZIURLSWUIHRB
|
7.0 | Kd | 57 | Yes | |
UIARLYUEJFELEN
|
6.8 | Kd | 289 | Yes | |
QNABDSWBQJKBHK
|
6.7 | IC50 | 45 | — | |
NHHQJBCNYHBUSI
|
6.4 | Kd | 220 | — | |
MFAQYJIYDMLAIM
|
6.4 | Kd | 130 | Yes | |
WPXVVAWAHQHJPF
|
6.3 | IC50 | 41 | — | |
OMZCMEYTWSXEPZ
|
6.2 | Kd | 43 | Yes | |
KTEIFNKAUNYNJU
|
6.2 | Kd | 114 | — | |
NXSJMRCTGYTSTK
|
6.1 | Kd | 200 | — | |
YYLKKYCXAOBSRM
|
6.1 | Kd | 191 | — | |
MVCOAUNKQVWQHZ
|
6.1 | Kd | 54 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |