Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDPXNCYWHLAZJC
|
6.3 | IC50 | 4 | — | |
SHKAUSIXYOWPKS
|
6.3 | IC50 | 3 | — | |
SJEYKCLWHCAMQL
|
6.3 | IC50 | 3 | — | |
SLWMPPADXCAMND
|
6.3 | IC50 | 3 | — | |
SMLYFAJYRKAOPL
|
6.3 | IC50 | 2 | — | |
SPUVKXRMQZAIAZ
|
6.3 | IC50 | 4 | — | |
SUWHOJVHZNVYPL
|
6.3 | IC50 | 2 | — | |
SYTDXYNETZANOI
|
6.3 | IC50 | 3 | — | |
SYYMSDGOIXLMBC
|
6.3 | IC50 | 3 | — | |
TZOPEIOUJFXKQZ
|
6.3 | IC50 | 3 | — | |
UIELDVYKNRNSEM
|
6.3 | IC50 | 3 | — | |
UKKBXHWKVGSVEV
|
6.3 | IC50 | 4 | — | |
UNVZWJFKXAEDKM
|
6.3 | IC50 | 2 | — | |
UQJWQNWEZPXTRQ
|
6.3 | IC50 | 3 | — | |
UUPSSROUZJUAGT
|
6.3 | IC50 | 2 | — | |
VATKWVNDCITFEB
|
6.3 | IC50 | 3 | — | |
VEIQGMIXACRMMO
|
6.3 | IC50 | 5 | — | |
VKRSAHZIVGFNMU
|
6.3 | IC50 | 2 | — | |
VPMFDTGNFBVOSP
|
6.3 | IC50 | 3 | — | |
VQRNHLREZMWHGF
|
6.3 | IC50 | 3 | — | |
VVDWMCFFRNYWGL
|
6.3 | IC50 | 3 | — | |
VWCXCYRYWPKZNG
|
6.3 | IC50 | 3 | — | |
VYVLFCZOKFCBJQ
|
6.3 | IC50 | 3 | — | |
WFNAULMUNPRODX
|
6.3 | IC50 | 2 | — | |
WGVZZDSXBCCRPN
|
6.3 | IC50 | 2 | — | |
WQHZIFFISAIJEF
|
6.3 | IC50 | 4 | — | |
WUCSNTVXKXMTBP
|
6.3 | IC50 | 3 | — | |
WVCAYXOTVLLXMU
|
6.3 | IC50 | 4 | — | |
WYZCWZRHCBLLRQ
|
6.3 | IC50 | 3 | — | |
XHBINYIIFGVWSM
|
6.3 | IC50 | 5 | — | |
XJAYAHAZZKYCJC
|
6.3 | IC50 | 3 | — | |
XRTAZINADDFLOG
|
6.3 | IC50 | 3 | — | |
XUCWVTDFYWWXFG
|
6.3 | IC50 | 3 | — | |
XXVRAEWUOFARHO
|
6.3 | IC50 | 3 | — | |
YETQQFMHUDZVIA
|
6.3 | IC50 | 5 | — | |
YNRDGUQMVYIVCM
|
6.3 | IC50 | 3 | — | |
YTGFCYJRAIFFGH
|
6.3 | IC50 | 4 | — | |
YXCHYSQVLDVUOJ
|
6.3 | IC50 | 3 | — | |
ZAMYFBONNUIDDG
|
6.3 | IC50 | 5 | — | |
ZBNFVHQEUFIFJM
|
6.3 | IC50 | 4 | — | |
ZCRLDBQMLFBFFN
|
6.3 | IC50 | 2 | — | |
ZDOPWPQLWDULEV
|
6.3 | IC50 | 3 | — | |
ZDTMGSSRQLKYTK
|
6.3 | IC50 | 5 | — | |
ZFGGQFYLMRFDEB
|
6.3 | IC50 | 3 | — | |
ZJWUMNUFLUTXRN
|
6.3 | IC50 | 2 | — | |
ZMGKRGOCDQRNTB
|
6.3 | IC50 | 3 | — | |
ZNKFCCNXFVRXHC
|
6.3 | IC50 | 3 | — | |
ZNOFYQJDWNDHAI
|
6.3 | IC50 | 4 | — | |
ZNTUEQOGCBDJQV
|
6.3 | IC50 | 2 | — | |
ZPDJVHLHIVCBBN
|
6.3 | IC50 | 3 | — |