Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KIHIMMDNUNDKTJ
|
6.3 | IC50 | 5 | — | |
KLDWSPPOKXJTIT
|
6.3 | IC50 | 4 | — | |
KNQFEIWYUMJEJW
|
6.3 | IC50 | 3 | — | |
KUIMRYDCYVFWRI
|
6.3 | IC50 | 2 | — | |
KURAWEFNNHDHOM
|
6.3 | IC50 | 3 | — | |
LDVUSEWLJKUPMB
|
6.3 | IC50 | 3 | — | |
LFVVFUDFYJQWPX
|
6.3 | IC50 | 3 | — | |
LHQPNVRFCKDYKG
|
6.3 | IC50 | 2 | — | |
LMPSDBKQPWYZFY
|
6.3 | IC50 | 3 | — | |
LNRUEHRMLQQRED
|
6.3 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
6.3 | Kd | 33 | Yes | |
LTXUQGNDYGUYMC
|
6.3 | IC50 | 3 | — | |
LUKFTCWBIWCAMK
|
6.3 | IC50 | 3 | — | |
MBKCHTMJAMAWPC
|
6.3 | IC50 | 5 | — | |
MBPRKKURYAKGON
|
6.3 | IC50 | 3 | — | |
MNDLFEMDUVUZEA
|
6.3 | IC50 | 2 | — | |
NAOSUZSDORYMKP
|
6.3 | IC50 | 3 | — | |
NHCXXCMLZIJGKZ
|
6.3 | IC50 | 3 | — | |
NJKVUYJCCZCQNK
|
6.3 | IC50 | 3 | — | |
NJQIBYWJBXKSRO
|
6.3 | IC50 | 5 | — | |
NJQIBYWJBXKSRO
|
6.3 | IC50 | 5 | — | |
NLASQQGOHZWAKY
|
6.3 | IC50 | 3 | — | |
NPSLABWCQNFJHJ
|
6.3 | IC50 | 5 | — | |
NQWKXHZZPBXKGF
|
6.3 | IC50 | 4 | — | |
NVKZQTWUWKWYCG
|
6.3 | IC50 | 3 | — | |
NYIGUQNAOHAUFR
|
6.3 | IC50 | 3 | — | |
OGAXAZKIMMCTIZ
|
6.3 | IC50 | 3 | — | |
OGNKTNDFGPEFFD
|
6.3 | IC50 | 3 | — | |
OUEOJFCFMCXADD
|
6.3 | IC50 | 4 | — | |
OZDWKTRNNHXKQT
|
6.3 | IC50 | 2 | — | |
PBZBHUPNRAUVJF
|
6.3 | IC50 | 2 | — | |
PFBDUGXDPNHKAM
|
6.3 | IC50 | 3 | — | |
PLTBBZBWBKAMPZ
|
6.3 | IC50 | 2 | — | |
PQYBSOBFELGWEF
|
6.3 | IC50 | 2 | — | |
PRVHVZIMFXZSQV
|
6.3 | IC50 | 3 | — | |
QFEUXSBOVSOXOY
|
6.3 | IC50 | 3 | — | |
QHBIMTBQLBHDHJ
|
6.3 | IC50 | 2 | — | |
QJMKYRIHQWAKSM
|
6.3 | IC50 | 3 | — | |
QKKRTUHQIAZEDD
|
6.3 | IC50 | 2 | — | |
QMONPAAOIIDBIL
|
6.3 | IC50 | 3 | — | |
QNPKKOXYJDZPQK
|
6.3 | IC50 | 2 | — | |
QPNYAXXXUXFKDG
|
6.3 | IC50 | 5 | — | |
QPQAGSRLQDSAGQ
|
6.3 | IC50 | 2 | — | |
QTWKCJAINLFWKV
|
6.3 | IC50 | 5 | — | |
RFKWUHOHGOAWTQ
|
6.3 | IC50 | 3 | — | |
RJGUQSMXHFQXPD
|
6.3 | IC50 | 3 | — | |
RNMZCDDYUSJWBE
|
6.3 | IC50 | 2 | — | |
RORFVUDLEIRGQY
|
6.3 | IC50 | 3 | — | |
RPLCLUCJTHAIOW
|
6.3 | IC50 | 3 | — | |
RZKGVOJSKFTTBA
|
6.3 | IC50 | 3 | — |