Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DGOBVCDUGLUZMU
|
6.3 | IC50 | 4 | — | |
DTMZOKHWEQAEJP
|
6.3 | IC50 | 4 | — | |
DTTUCRMZJFXMJK
|
6.3 | IC50 | 3 | — | |
DYYJQOFBFXWRDD
|
6.3 | IC50 | 3 | — | |
FAJVOBZBVGQKFD
|
6.3 | IC50 | 3 | — | |
FGHXOSBHGQKMBX
|
6.3 | IC50 | 4 | — | |
FIJYWRPWHKFPLQ
|
6.3 | IC50 | 3 | — | |
FJUIAQIBGJSIJS
|
6.3 | IC50 | 3 | — | |
FRHNEIRUMPIDKL
|
6.3 | IC50 | 3 | — | |
FSJDACURTSWGHC
|
6.3 | IC50 | 3 | — | |
FSJDACURTSWGHC
|
6.3 | IC50 | 5 | — | |
FSJDACURTSWGHC
|
6.3 | IC50 | 4 | — | |
FSNXDZZUWFZSPA
|
6.3 | IC50 | 3 | — | |
FTIMKXNADWOPKE
|
6.3 | IC50 | 3 | — | |
FYJMEEVVSSJUMQ
|
6.3 | IC50 | 4 | — | |
FZGGLLMOLZVRHY
|
6.3 | IC50 | 3 | — | |
GAKPIAPJVGZESM
|
6.3 | IC50 | 4 | — | |
GBVHHGINCYVVRZ
|
6.3 | IC50 | 2 | — | |
GCBUMMPSFVNQKY
|
6.3 | IC50 | 2 | — | |
GKDGCIISLGIYBM
|
6.3 | IC50 | 3 | — | |
GNBFLDHHHUBBFG
|
6.3 | IC50 | 3 | — | |
GOTKNVOMZNDPKT
|
6.3 | IC50 | 3 | — | |
GYWNYPUPJODCTA
|
6.3 | IC50 | 3 | — | |
HAVVSQSFGAQFOW
|
6.3 | IC50 | 2 | — | |
HJOMYFVOXGNASK
|
6.3 | IC50 | 2 | — | |
HLDHNATWCDWAML
|
6.3 | IC50 | 3 | — | |
HMNGFRURISAKFO
|
6.3 | IC50 | 3 | — | |
HQHKCYQAKIHFNI
|
6.3 | IC50 | 3 | — | |
HSVSYWHNTHEXTN
|
6.3 | IC50 | 3 | — | |
HTKJGEPLONIJLG
|
6.3 | IC50 | 3 | — | |
HVXKQKFEHMGHSL
|
6.3 | IC50 | 5 | — | |
HZOGQCYCMSFESW
|
6.3 | IC50 | 4 | — | |
IFVXCNKRSUKURE
|
6.3 | IC50 | 4 | — | |
IIBGPAMZGFHRRY
|
6.3 | IC50 | 2 | — | |
INTICWGTKLQPSH
|
6.3 | IC50 | 3 | — | |
IOXJGKZLPLFOBF
|
6.3 | IC50 | 5 | — | |
IQEZRSQHZBKCOU
|
6.3 | IC50 | 4 | — | |
IUKSUNXUYRVVIQ
|
6.3 | IC50 | 3 | — | |
IVTMGIFJCKLZRO
|
6.3 | IC50 | 3 | — | |
IXLSYYGZAKKXCH
|
6.3 | IC50 | 3 | — | |
JFLJVHMCZLMBSN
|
6.3 | IC50 | 3 | — | |
JFXUNTVGMAFDCX
|
6.3 | IC50 | 3 | — | |
JJQTYTQYXOULRB
|
6.3 | IC50 | 5 | — | |
JOGJAGGMXRVDDM
|
6.3 | IC50 | 2 | — | |
JVJKGDUZNRRKIX
|
6.3 | IC50 | 3 | — | |
KBVAWHBMEYHTMD
|
6.3 | IC50 | 3 | — | |
KCGTXHCPPMDHIJ
|
6.3 | IC50 | 3 | — | |
KCIJBEJQKOVUTG
|
6.3 | IC50 | 3 | — | |
KDAFZLQNEAKVCC
|
6.3 | IC50 | 5 | — | |
KHSJGHHCLKKKKU
|
6.3 | IC50 | 5 | — |